SCHEMBL30587482

SCHEMBL30587482

O=C(O)c1nc2cccc(-c3ccccc3)c2s1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 1/20 0.47
HNF4A P41235 1/20 0.45
ASH1L Q9NR48 1/20 0.42
SMN1; SMN2 Q16637 4/20 0.41
NPC1 O15118 2/20 0.41
NFKB1 P19838 2/20 0.41
RAB9A P51151 2/20 0.41
NFKB2 Q00653 2/20 0.41
RELA Q04206 2/20 0.41
PKM P14618 1/20 0.41
DHODH Q02127 2/20 0.40
PDE10A Q9Y233 2/20 0.40
HDAC1 Q13547 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
RET P07949 1/20 0.39
FLT1 P17948 1/20 0.39
KDR P35968 1/20 0.39
MAPK14 Q16539 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18366688 1.00 RIPK1 (0.47) RIPK1HNF4AASH1LSMN1; SMN2NPC1
SCHEMBL19659306 0.88 RIPK1 (0.46) RIPK1ASH1LSMN1; SMN2NPC1NFKB1
SCHEMBL30587519 0.77 AKR1B1 (0.42) SMN1; SMN2NPC1NFKB1RAB9ANFKB2
SCHEMBL7960065 0.77 AKR1A1 (0.43) RIPK1SMN1; SMN2NPC1NFKB1RAB9A
SCHEMBL14860945 0.75 ASH1L (0.62) ASH1LNPC1NFKB1RAB9ANFKB2
SCHEMBL31621268 0.75 ASH1L (0.62) ASH1LNPC1NFKB1RAB9ANFKB2
SCHEMBL836745 0.72 SMN1; SMN2 (0.65) SMN1; SMN2NPC1NFKB1RAB9ANFKB2
SCHEMBL28727291 0.72 SMN1; SMN2 (0.65) SMN1; SMN2NPC1NFKB1RAB9ANFKB2
SCHEMBL6068377 0.71 NPC1 (0.64) SMN1; SMN2NPC1RAB9A
Hydrochloric Acid SCHEMBL3610419 0.70 SMN1; SMN2 (0.63) SMN1; SMN2NPC1NFKB1RAB9ANFKB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111269221-B Bicyclic lactams and methods of use thereof 豪夫迈·罗氏有限公司 2023-09-26 CN disclosed