SCHEMBL30593285

SCHEMBL30593285

NC(=O)N1CCc2ccccc2C1c1coc2ccccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 2/20 0.43
SLC6A2 P23975 1/20 0.43
SLC6A3 Q01959 1/20 0.43
CHRNB2 P17787 1/20 0.40
CHRNA4 P43681 1/20 0.40
ACE P12821 2/20 0.39
CHRM3 P20309 3/20 0.39
CACNA1F O60840 1/20 0.39
CHRM2 P08172 1/20 0.39
CHRM4 P08173 1/20 0.39
CHRM5 P08912 1/20 0.39
CHRM1 P11229 1/20 0.39
KCNE1 P15382 1/20 0.39
KCNQ1 P51787 1/20 0.39
CACNA1D Q01668 1/20 0.39
KCNH2 Q12809 1/20 0.39
CACNA1S Q13698 1/20 0.39
CACNA1C Q13936 1/20 0.39
SCN5A Q14524 1/20 0.39
KCND3 Q9UK17 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31070630 0.88 SLC6A4 (0.50) SLC6A4SLC6A2SLC6A3CHRNB2CHRNA4
SCHEMBL30593239 0.86 DRD2 (0.41) CHRNB2CHRNA4DRD2
SCHEMBL25604564 0.76 HHAT (0.57) CHRM3CACNA1FCHRM2CHRM4CHRM5
SCHEMBL31070610 0.76 DRD2 (0.38) SLC6A4SLC6A2SLC6A3CHRNB2CHRNA4
SCHEMBL30593289 0.76 LMNA (0.43) SLC6A4CHRM3CACNA1FCHRM2CHRM4
SCHEMBL30593300 0.76 DRD2 (0.49) DRD2
SCHEMBL29084782 0.73 DRD1 (0.43) CHRM3HDAC3HDAC1HDAC2HDAC8
SCHEMBL30593320 0.72 CHRM3 (0.45) CHRM3KCNH2HDAC3HDAC1HDAC2
SCHEMBL31070552 0.72 SLC6A4 (0.47) SLC6A4SLC6A2SLC6A3CHRNB2CHRNA4
SCHEMBL30965951 0.72 TRPM8 (0.60) CHRM3KCNH2HHATTRPM8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118742543-A Dihydro isoquinoline compound and medical application thereof 中国科学院上海药物研究所 2024-10-01 CN disclosed
CN-116789641-A Dihydro isoquinoline compound and medical application thereof 中国科学院上海药物研究所 2023-09-22 CN disclosed