SCHEMBL30593289

SCHEMBL30593289

NC(=O)N1CCc2ccccc2C1c1csc2ccccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.43
MAPT P10636 1/20 0.43
HHAT Q5VTY9 2/20 0.39
CHRM3 P20309 4/20 0.39
CACNA1F O60840 1/20 0.39
CHRM2 P08172 1/20 0.39
CHRM4 P08173 1/20 0.39
CHRM5 P08912 1/20 0.39
CHRM1 P11229 1/20 0.39
KCNE1 P15382 1/20 0.39
KCNQ1 P51787 1/20 0.39
CACNA1D Q01668 1/20 0.39
KCNH2 Q12809 1/20 0.39
CACNA1S Q13698 1/20 0.39
CACNA1C Q13936 1/20 0.39
SCN5A Q14524 1/20 0.39
KCND3 Q9UK17 1/20 0.39
DPP4 P27487 1/20 0.39
DPP8 Q6V1X1 1/20 0.39
DPP9 Q86TI2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31070553 0.88 MAPT (0.39) LMNAMAPTKCNH2DPP4DPP8
SCHEMBL25604564 0.76 HHAT (0.57) HHATCHRM3CACNA1FCHRM2CHRM4
SCHEMBL30593285 0.76 SLC6A4 (0.43) HHATCHRM3CACNA1FCHRM2CHRM4
SCHEMBL30593300 0.76 DRD2 (0.49) LMNAMAPTDRD2
SCHEMBL29084782 0.73 DRD1 (0.43) LMNAMAPTHHATCHRM3HDAC3
SCHEMBL31070488 0.73 MEN1 (0.39) LMNAMAPTHDAC8DRD2SLC6A4
SCHEMBL30593320 0.72 CHRM3 (0.45) CHRM3KCNH2HDAC3HDAC1HDAC2
SCHEMBL30965951 0.72 TRPM8 (0.60) HHATCHRM3KCNH2
SCHEMBL17559775 0.72 TRPM8 (0.57) HHAT
SCHEMBL30965925 0.72 TRPM8 (0.60) HHATCHRM3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118742543-A Dihydro isoquinoline compound and medical application thereof 中国科学院上海药物研究所 2024-10-01 CN disclosed
CN-116789641-A Dihydro isoquinoline compound and medical application thereof 中国科学院上海药物研究所 2023-09-22 CN disclosed