SCHEMBL30656350

SCHEMBL30656350

Cc1ncsc1COc1ccc2sc(C)c(C(=O)NC3(CO)CCC3)c2c1

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 3/20 0.34
ABL1 P00519 1/20 0.34
CNR2 P34972 6/20 0.33
EGLN2 Q96KS0 2/20 0.33
EGLN1 Q9GZT9 2/20 0.33
CNR1 P21554 2/20 0.33
KMT2A Q03164 1/20 0.33
ESR1 P03372 1/20 0.32
ESR2 Q92731 1/20 0.32
ALDH1A1 P00352 1/20 0.31
SCN9A Q15858 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
ADAMTS4 O75173 1/20 0.30
MMP3 P08254 1/20 0.30
MMP7 P09237 1/20 0.30
ADAMTS1 Q9UHI8 1/20 0.30
ADAMTS5 Q9UNA0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30656026 0.96 SCN9A (0.33) ADAM17KMT2AESR1ESR2ALDH1A1
SCHEMBL30656018 0.92 ADAM17 (0.38) ADAM17CNR2EGLN2EGLN1CNR1
SCHEMBL30655952 0.91 ADAM17 (0.32) ADAM17ESR1ESR2L3MBTL1ADAMTS4
SCHEMBL24485585 0.84 GAA (0.43) KMT2AALDH1A1L3MBTL1
SCHEMBL29630101 0.84 GAA (0.43) KMT2AALDH1A1L3MBTL1
SCHEMBL30656104 0.83 ABL1 (0.36) ADAM17ABL1CNR2CNR1KMT2A
SCHEMBL30656117 0.83 MEN1 (0.37) KMT2AESR1ESR2L3MBTL1
SCHEMBL30656008 0.82 MAPK14 (0.38) ADAM17CNR2KMT2A
SCHEMBL30656103 0.82 SLC6A5 (0.43)
SCHEMBL24485388 0.80 GAA (0.44) KMT2AALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250346569-A1 NEW DERIVATIVES FOR TREATING TRPM3 MEDIATED DISORDERS UNIV LEUVEN KATH (BE) 2025-11-13 US claimed
EP-4532013-A1 NEW DERIVATIVES FOR TREATING TRPM3 MEDIATED DISORDERS Katholieke Universiteit Leuven KU Leuven Research & Development (BE) 2025-04-09 EP claimed
CN-119421879-A Novel derivatives for the treatment of TRPM3 mediated disorders 勒芬天主教大学 2025-02-11 CN claimed
WO-2023227697-A1 NEW DERIVATIVES FOR TREATING TRPM3 MEDIATED DISORDERS KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2023-11-30 WO claimed
US-20250346569-A1 NEW DERIVATIVES FOR TREATING TRPM3 MEDIATED DISORDERS UNIV LEUVEN KATH (BE) 2025-11-13 US disclosed
EP-4532013-A1 NEW DERIVATIVES FOR TREATING TRPM3 MEDIATED DISORDERS Katholieke Universiteit Leuven KU Leuven Research & Development (BE) 2025-04-09 EP disclosed
CN-119421879-A Novel derivatives for the treatment of TRPM3 mediated disorders 勒芬天主教大学 2025-02-11 CN disclosed
WO-2023227697-A1 NEW DERIVATIVES FOR TREATING TRPM3 MEDIATED DISORDERS KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2023-11-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250346569-A1 NEW DERIVATIVES FOR TREATING TRPM3 MEDIATED DISORDERS TRPM4, TRPM2, TRPM6 ADAM17 2628/4885ABL1 4202/4885CNR2 100/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.