SCHEMBL3066433

SCHEMBL3066433

NC(=O)C[C@H](O)C(=O)N1CC[C@@H](O)C1

nearest known ligand 0.51

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 12/20 0.51
DPP7 Q9UHL4 9/20 0.51
DPP8 Q6V1X1 4/20 0.35
DPP9 Q86TI2 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21548468 0.83 DPP7 (0.63) DPP4DPP7DPP8DPP9
SCHEMBL3066436 0.81 DPP7 (0.60) DPP4DPP7DPP8DPP9
SCHEMBL5789549 0.75 DPP7 (0.66) DPP4DPP7DPP8DPP9
SCHEMBL5789775 0.75 DPP7 (0.66) DPP4DPP7DPP8DPP9
SCHEMBL10311720 0.74 DPP4 (0.60) DPP4DPP7DPP8DPP9
SCHEMBL738423 0.74 DPP4 (0.60) DPP4DPP7DPP8DPP9
SCHEMBL10311683 0.74 DPP4 (0.60) DPP4DPP7DPP8DPP9
SCHEMBL3067845 0.74 DPP7 (0.43) DPP4DPP7
SCHEMBL12801567 0.73 DPP4 (0.58) DPP4DPP7DPP8DPP9
SCHEMBL12801568 0.73 DPP4 (0.58) DPP4DPP7DPP8DPP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100267719-A1 Enhanced Indolinone Based Protein Kinase Inhibitors THE SCRIPPS RESEARCH INSTITUTE (US) 2010-10-21 US disclosed
EP-1893194-A4 ENHANCED INDOLINONE BASED PROTEIN KINASE INHIBITORS SCRIPPS RESEARCH INST (US) 2009-07-01 EP disclosed
EP-1893194-A1 ENHANCED INDOLINONE BASED PROTEIN KINASE INHIBITORS The Scripps Research Institute (US) 2008-03-05 EP disclosed
US-20060287381-A1 Enhanced indolinone based protein kinase inhibitors THE SCRIPPS RESEARCH INSTITUTE (US) 2006-12-21 US disclosed
WO-2006127961-A1 ENHANCED INDOLINONE BASED PROTEIN KINASE INHIBITORS THE SCRIPPS RESEARCH INSTITUTE (US) 2006-11-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060287381-A1 Enhanced indolinone based protein kinase inhibitors PHKG1, PHKG2, PRKCH DPP4 2943/4885DPP7 2012/4885DPP8 2558/4885
US-20100267719-A1 Enhanced Indolinone Based Protein Kinase Inhibitors PHKG1, PHKG2, PRKCH DPP4 3646/4885DPP7 2387/4885DPP8 2930/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.