SCHEMBL30679697

SCHEMBL30679697

Nc1cccc(N)c1-c1ncncn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 2/20 0.42
CYP3A4 P08684 6/20 0.36
TSHR P16473 4/20 0.36
ALDH1A1 P00352 4/20 0.36
HSD17B10 Q99714 3/20 0.36
HPGD P15428 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
CASP1 P29466 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
ALOX15 P16050 1/20 0.35
CASP7 P55210 1/20 0.35
PIK3CA P42336 1/20 0.35
PTPRC P08575 1/20 0.34
ADORA2A P29274 1/20 0.34
LMNA P02545 2/20 0.33
CYP2D6 P10635 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
EGFR P00533 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9704689 0.85 HSP90AA1 (0.46) HSP90AA1TSHRALDH1A1HSD17B10HPGD
SCHEMBL22232393 0.80 ADRB2 (0.41) HSP90AA1CYP3A4TSHRALDH1A1HSD17B10
SCHEMBL14314286 0.80 PARP1 (0.40) TSHRALDH1A1HSD17B10HPGDKEAP1
SCHEMBL28604840 0.78 HSP90AA1 (0.43) HSP90AA1CYP3A4EGFR
SCHEMBL12452253 0.76 NOS3 (0.38) HSP90AA1CYP3A4TSHRALDH1A1HPGD
SCHEMBL1317752 0.76 ALDH1A1 (0.37) HSP90AA1CYP3A4TSHRALDH1A1HSD17B10
SCHEMBL14314312 0.75 PLK1 (0.41) ALDH1A1HSD17B10HPGDLMNACYP2C9
SCHEMBL29889875 0.74 ALDH1A1 (0.52) HSP90AA1CYP3A4ALDH1A1HSD17B10HPGD
SCHEMBL6565668 0.74 ALDH1A1 (0.52) HSP90AA1CYP3A4ALDH1A1HSD17B10HPGD
SCHEMBL29521927 0.74 ALDH1A1 (0.52) HSP90AA1CYP3A4TSHRALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117430600-A Selective EGFR inhibitor, preparation method and pharmaceutical application thereof 上海和誉生物医药科技有限公司 2024-01-23 CN disclosed