SCHEMBL30689233

SCHEMBL30689233

CN(CC(=O)Nc1cc[nH]c(=O)c1N)C(=O)OCc1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PRSS1 P07477 1/20 0.45
TPSAB1 Q15661 1/20 0.45
CACNA1H O95180 4/20 0.41
ROCK2 O75116 3/20 0.41
HDAC1 Q13547 1/20 0.40
ABCB1 P08183 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.37
CDC42 P60953 1/20 0.37
ROCK1 Q13464 1/20 0.37
PKN2 Q16513 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
F13A1 P00488 1/20 0.37
TGM2 P21980 1/20 0.37
TGM1 P22735 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7336752 0.76 SHMT2 (0.51) PRSS1TPSAB1CACNA1HHDAC1L3MBTL1
SCHEMBL8426730 0.74 PRSS1 (0.56) PRSS1TPSAB1CACNA1HABCB1L3MBTL1
SCHEMBL855297 0.73 HDAC1 (0.47) PRSS1TPSAB1CACNA1HHDAC1NPC1
SCHEMBL29940493 0.72 PRSS1 (0.41) PRSS1TPSAB1CACNA1HHDAC1NPC1
SCHEMBL29302722 0.72 PRSS1 (0.41) PRSS1TPSAB1CACNA1HHDAC1NPC1
SCHEMBL11517533 0.71 PRSS1 (0.60) PRSS1TPSAB1CACNA1HABCB1RAB9A
SCHEMBL8571304 0.71 PRSS1 (0.63) PRSS1TPSAB1CACNA1HHDAC1ABCB1
SCHEMBL5331588 0.71 ALDH1A1 (0.51) PRSS1TPSAB1ABCB1L3MBTL1F13A1
SCHEMBL8241799 0.70 CACNA1H (0.56) PRSS1TPSAB1CACNA1HABCB1F13A1
SCHEMBL7505433 0.70 PRSS1 (0.59) PRSS1TPSAB1CACNA1HABCB1F13A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023250157-A9 INHIBITORS OF MYCOBACTERIUM TUBERCULOSIS LIPOAMIDE DEHYDROGENASE CORNELL UNIVERSITY (US) 2024-01-25 WO disclosed
WO-2023250157-A1 INHIBITORS OF MYCOBACTERIUM TUBERCULOSIS LIPOAMIDE DEHYDROGENASE CORNELL UNIVERSITY (US) 2023-12-28 WO disclosed