SCHEMBL30712604

SCHEMBL30712604

[2H]C1([2H])OC(=O)NC1c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
BRD4 O60885 1/20 0.36
KMT2A Q03164 3/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35
GFER P55789 1/20 0.35
HSD17B10 Q99714 1/20 0.35
MEN1 O00255 2/20 0.34
PRCP P42785 1/20 0.34
LMNA P02545 2/20 0.34
CYP19A1 P11511 1/20 0.34
NPC1 O15118 1/20 0.34
ADORA3 P0DMS8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30712598 1.00 CA2 (0.38) CA2SMN1; SMN2BRD4KMT2AKDM4E
SCHEMBL30712600 0.82 TDP1 (0.42) SMN1; SMN2KMT2AKDM4EALDH1A1GAA
SCHEMBL30712573 0.82 TDP1 (0.42) SMN1; SMN2KMT2AKDM4EALDH1A1GAA
SCHEMBL445133 0.81 SMN1; SMN2 (0.42) CA2SMN1; SMN2BRD4KMT2AKDM4E
SCHEMBL4563 0.81 SMN1; SMN2 (0.42) CA2SMN1; SMN2BRD4KMT2AKDM4E
SCHEMBL4562 0.81 SMN1; SMN2 (0.42) CA2SMN1; SMN2BRD4KMT2AKDM4E
SCHEMBL16106147 0.81 SMN1; SMN2 (0.42) CA2SMN1; SMN2BRD4KMT2AKDM4E
SCHEMBL2909384 0.79 AR (0.41) CA2SMN1; SMN2BRD4KMT2AALDH1A1
SCHEMBL5031878 0.78 CA2 (0.38) CA2SMN1; SMN2BRD4KMT2AKDM4E
SCHEMBL14831166 0.71 TAAR1 (0.41) BRD4KMT2AKDM4EALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119790041-A Alpha, beta-unsaturated amide compounds, preparation method, pharmaceutical composition and application thereof 中国科学院上海药物研究所 2025-04-08 CN disclosed
CN-117402123-A Alpha, beta-unsaturated amide compounds, preparation method, pharmaceutical composition and application thereof 中国科学院上海药物研究所 2024-01-16 CN disclosed
WO-2024008166-A1 α,β-UNSATURATED AMIDE COMPOUND, AND PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL COMPOSITION AND USE THEREOF 中国科学院上海药物研究所 2024-01-11 WO disclosed