SCHEMBL30713271

SCHEMBL30713271

COC(=O)C(=O)NCc1ncc(Br)cc1Cl

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.36
HPGD P15428 2/20 0.36
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
LMNA P02545 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
PLAU P00749 1/20 0.34
GPR35 Q9HC97 1/20 0.34
TET2 Q6N021 1/20 0.33
EGLN1 Q9GZT9 1/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
ROCK2 O75116 1/20 0.33
ROCK1 Q13464 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
RECQL P46063 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29277569 1.00 TSHR (0.36) TSHRHPGDNPC1RAB9ALMNA
SCHEMBL27389799 0.88 GPR35 (0.49) TSHRHPGDNPC1RAB9ASMN1; SMN2
SCHEMBL30357636 0.88 GPR35 (0.49) TSHRHPGDNPC1RAB9ASMN1; SMN2
SCHEMBL31481925 0.84 GPR35 (0.38) TSHRHPGDNPC1RAB9ASMN1; SMN2
SCHEMBL16793840 0.81 NPC1 (0.39) TSHRNPC1RAB9ALMNASMN1; SMN2
SCHEMBL16809853 0.78 AAK1 (0.45) LMNAKDM4E
SCHEMBL30162902 0.78 AAK1 (0.45) LMNAKDM4E
SCHEMBL18335081 0.77 LMNA (0.41) TSHRHPGDNPC1RAB9ALMNA
SCHEMBL29277634 0.72 SMN1; SMN2 (0.41) TSHRNPC1RAB9ASMN1; SMN2KMT2A
SCHEMBL30713233 0.72 SMN1; SMN2 (0.41) TSHRNPC1RAB9ASMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117304183-A Five-membered and six-membered nitrogen-containing compound, intermediate thereof, preparation method and application 杭州圣域生物医药科技有限公司 2023-12-29 CN disclosed