SCHEMBL30714632

SCHEMBL30714632

Cc1ncc(COc2ccc3nn(C)c(C(=O)N[C@@H](CO)C(N)=O)c3c2)s1

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.33
MCHR1 Q99705 3/20 0.33
L3MBTL1 Q9Y468 1/20 0.32
SCN9A Q15858 2/20 0.31
NPC1 O15118 3/20 0.31
RAB9A P51151 3/20 0.31
GUCY1B2 O75343 1/20 0.31
GUCY1A2 P33402 1/20 0.31
GUCY1A1 Q02108 1/20 0.31
GUCY1B1 Q02153 1/20 0.31
POLB P06746 1/20 0.31
PDE10A Q9Y233 1/20 0.30
CNR1 P21554 1/20 0.30
CNR2 P34972 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30714669 0.90 HPGDS (0.38) KMT2AMCHR1L3MBTL1SCN9ANPC1
SCHEMBL30714744 0.90 HPGDS (0.38) KMT2AMCHR1L3MBTL1SCN9ANPC1
SCHEMBL30714634 0.87 KMT2A (0.34) KMT2AMCHR1L3MBTL1SCN9ANPC1
SCHEMBL30714683 0.84 NPC1 (0.34) KMT2ASCN9ANPC1RAB9APOLB
SCHEMBL30714617 0.83 CYP11B2 (0.37) KMT2AL3MBTL1SCN9ANPC1RAB9A
SCHEMBL30714605 0.83 KLKB1 (0.33) KMT2AMCHR1SCN9ANPC1RAB9A
SCHEMBL30714691 0.83 KLKB1 (0.33) KMT2AMCHR1SCN9ANPC1RAB9A
SCHEMBL30714604 0.82 MCHR1 (0.37) KMT2AMCHR1L3MBTL1NPC1RAB9A
SCHEMBL30714670 0.82 MCHR1 (0.40) KMT2AMCHR1L3MBTL1NPC1RAB9A
SCHEMBL26874836 0.82 MCHR1 (0.37) KMT2AMCHR1L3MBTL1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250376461-A1 INDAZOLE DERIVATIVES FOR TREATING TRPM3-MEDIATED DISORDERS UNIV LEUVEN KATH (BE) 2025-12-11 US disclosed
EP-4499624-A2 INDAZOLE DERIVATIVES FOR TREATING TRPM3-MEDIATED DISORDERS Katholieke Universiteit Leuven KU Leuven Research & Development (BE) 2025-02-05 EP disclosed
WO-2023230540-A2 INDAZOLE DERIVATIVES FOR TREATING TRPM3-MEDIATED DISORDERS KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2023-11-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250376461-A1 INDAZOLE DERIVATIVES FOR TREATING TRPM3-MEDIATED DISORDERS TRPV3, TRPM2, TRPV1 KMT2A 3017/4885MCHR1 1891/4885L3MBTL1 4209/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.