SCHEMBL3071652

SCHEMBL3071652

Nc1ccc2c(c1Br)C(O)CC2

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL585157 0.77 CYP11B1 (0.35)
SCHEMBL3067329 0.74 EPAS1 (0.35)
SCHEMBL4643692 0.73 ALDH1A1 (0.38)
SCHEMBL27455229 0.70 HTR2A (0.40)
SCHEMBL18986893 0.69 P2RX7 (0.37)
SCHEMBL31722382 0.69 P2RX7 (0.37)
SCHEMBL17397762 0.69 P2RX7 (0.37)
SCHEMBL12584160 0.69 P2RX7 (0.37)
SCHEMBL4819283 0.68 EPAS1 (0.33)
SCHEMBL22012098 0.65 PARP1 (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8399490-B2 Insecticides SYNGENTA CROP PROTECTION LLC (US) 2013-03-19 US disclosed
US-20100273830-A1 NOVEL INSECTICIDES SYNGENTA CROP PROTECTION, INC. (US) 2010-10-28 US disclosed
CN-101743237-A condensed anthranilamide insecticides SYNGENTA PARTICIPATIONS AG 2010-06-16 CN disclosed
EP-2167484-A2 CONDENSED ANTHRANILAMIDE INSECTICIDES Syngeta Participations AG (CH) 2010-03-31 EP disclosed
WO-2009010260-A2 CONDENSED ANTHRANILAMIDE INSECTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2009-01-22 WO disclosed