SCHEMBL30718239

SCHEMBL30718239

c1ccc2ncc(-c3ccnc(N4CCNCC4)n3)cc2c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.53
CHRNA4 P43681 1/20 0.53
DKK1 O94907 2/20 0.49
NISCH Q9Y2I1 1/20 0.47
ADRB1 P08588 1/20 0.45
MYLK4 Q86YV6 3/20 0.45
STK17A Q9UEE5 3/20 0.45
MAPKAPK2 P49137 1/20 0.45
ACHE P22303 3/20 0.44
PIK3CA P42336 2/20 0.44
ALDH1A1 P00352 2/20 0.44
PIK3CD O00329 1/20 0.44
PIK3R1 P27986 1/20 0.44
PIK3CB P42338 1/20 0.44
KDM4E B2RXH2 1/20 0.44
PDGFRB P09619 1/20 0.43
PDGFRA P16234 1/20 0.43
CLK4 Q9HAZ1 1/20 0.43
TBK1 Q9UHD2 1/20 0.43
HPGD P15428 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27029440 1.00 CHRNB2 (0.53) CHRNB2CHRNA4DKK1NISCHADRB1
SCHEMBL27063740 0.95 CHRNB2 (0.61) CHRNB2CHRNA4DKK1NISCHADRB1
SCHEMBL29931680 0.87 DKK1 (0.51) CHRNB2CHRNA4DKK1NISCHPIK3CA
SCHEMBL27029515 0.85 HTR3A (0.58) DKK1STK17AACHEPIK3CAKDM4E
SCHEMBL30718191 0.85 HTR3A (0.58) DKK1STK17AACHEPIK3CAKDM4E
SCHEMBL29931584 0.84 DKK1 (0.51) CHRNB2CHRNA4DKK1NISCHPIK3CA
SCHEMBL3652486 0.83 DKK1 (0.69) DKK1ADRB1MYLK4STK17AACHE
SCHEMBL27029497 0.83 DKK1 (0.72) DKK1PIK3CAPIK3CDPIK3R1PIK3CB
SCHEMBL30718212 0.83 CHRNB2 (0.51) CHRNB2CHRNA4NISCHADRB1PIK3CA
SCHEMBL27029561 0.83 CHRNB2 (0.51) CHRNB2CHRNA4NISCHADRB1PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117157284-A CTLA-4 small molecule degradation agent and application thereof 苏州国匡医药科技有限公司 2023-12-01 CN disclosed