SCHEMBL6237782

SCHEMBL6237782

COc1ccccc1Nc1nc(Cl)nc(Cl)n1

nearest known ligand 0.93

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.93
ALDH1A1 P00352 5/20 0.93
KMT2A Q03164 2/20 0.93
KDM4E B2RXH2 1/20 0.93
SMN1; SMN2 Q16637 1/20 0.93
NPSR1 Q6W5P4 1/20 0.76
TSHR P16473 2/20 0.61
GAA P10253 3/20 0.60
NPC1 O15118 2/20 0.57
RAB9A P51151 2/20 0.57
L3MBTL1 Q9Y468 2/20 0.57
LRRK2 Q5S007 1/20 0.57
EGFR P00533 1/20 0.56
POLB P06746 1/20 0.51
PTK2 Q05397 1/20 0.51
GBA1 P04062 2/20 0.50
NFKB1 P19838 1/20 0.50
THRB P10828 1/20 0.49
USP2 O75604 1/20 0.49
MEN1 O00255 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29609022 1.00 MAPT (0.93) MAPTALDH1A1KMT2AKDM4ESMN1; SMN2
SCHEMBL28939641 0.91 MAPT (0.88) MAPTALDH1A1KMT2AKDM4ESMN1; SMN2
Dyrene SCHEMBL8178116 0.89 TSHR (0.75) MAPTALDH1A1KMT2AKDM4ESMN1; SMN2
SCHEMBL11813903 0.87 MAPT (0.83) MAPTALDH1A1KMT2AKDM4ESMN1; SMN2
Dyrene SCHEMBL1029356 0.82 MAPT (0.65) MAPTALDH1A1KMT2AKDM4ESMN1; SMN2
SCHEMBL13326002 0.81 MAPT (0.71) MAPTALDH1A1KMT2AKDM4ESMN1; SMN2
SCHEMBL11837274 0.81 TSHR (0.80) MAPTALDH1A1KMT2AKDM4ESMN1; SMN2
Dyrene SCHEMBL5954767 0.81 TSHR (0.86) MAPTALDH1A1KMT2AKDM4ESMN1; SMN2
SCHEMBL28176767 0.80 MAPT (0.65) MAPTALDH1A1KMT2AKDM4ESMN1; SMN2
SCHEMBL9697643 0.79 MAPT (0.66) MAPTALDH1A1KMT2AKDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108191774-B Heterocyclic compound, preparation method and application thereof 中国药科大学 2022-05-24 CN disclosed
US-7718655-B2 Trisubstituted triazine compounds, and methods for making and using the compounds, which have antitubulin activity NEW YORK UNIVERSITY (US) 2010-05-18 US disclosed
US-7718655-B2 Trisubstituted triazine compounds, and methods for making and using the compounds, which have antitubulin activity NEW YORK UNIVERSITY (US) 2010-05-18 US disclosed
WO-2005011703-A1 2-CYANO-1,3,5-TRIAZINE-4,6-DIAMINE DERIVATIVES AKZO NOBEL N.V. (NL) 2005-02-10 WO disclosed