Predicted protein targets (top 20)
| gene | UniProt | supporting neighbours | confidence | |
|---|---|---|---|---|
| ▸ | GRM8 | O00222 | 2/20 | 0.62 |
| ▸ | GRM6 | O15303 | 2/20 | 0.62 |
| ▸ | GRM7 | Q14831 | 2/20 | 0.62 |
| ▸ | GRM4 | Q14833 | 2/20 | 0.62 |
| ▸ | GSR | P00390 | 2/20 | 0.62 |
| ▸ | GRIN2D | O15399 | 1/20 | 0.62 |
| ▸ | GRIN3B | O60391 | 1/20 | 0.62 |
| ▸ | CYP1A2 | P05177 | 1/20 | 0.62 |
| ▸ | GRIK1 | P39086 | 1/20 | 0.62 |
| ▸ | GRM5 | P41594 | 1/20 | 0.62 |
| ▸ | GRIA1 | P42261 | 1/20 | 0.62 |
| ▸ | GRIA2 | P42262 | 1/20 | 0.62 |
| ▸ | GRIA3 | P42263 | 1/20 | 0.62 |
| ▸ | SLC1A3 | P43003 | 1/20 | 0.62 |
| ▸ | SLC1A2 | P43004 | 1/20 | 0.62 |
| ▸ | SLC1A1 | P43005 | 1/20 | 0.62 |
| ▸ | GRIA4 | P48058 | 1/20 | 0.62 |
| ▸ | GRIN1 | Q05586 | 1/20 | 0.62 |
| ▸ | GRIN2A | Q12879 | 1/20 | 0.62 |
| ▸ | GRIK2 | Q13002 | 1/20 | 0.62 |
Click a target to see other patent compounds predicted against it — the reverse direction, in place.
Similar compounds — the chemically nearest patent molecules
Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.
| Compound | similarity | top predicted | shared targets | |
|---|---|---|---|---|
| Glutamine SCHEMBL9716039 | 0.88 | ALOX15 (0.63) | GRM8GRM6GRM7GRM4GSR | |
| Glycine SCHEMBL8588130 | 0.87 | GLRA1 (0.42) | GRM8GRM6GRM7GRM4GSR | |
| SCHEMBL352049 | 0.87 | SLC1A5 (0.43) | GRM8GRM6GRM7GRM4GSR | |
| SCHEMBL3502798 | 0.87 | SLC1A5 (0.43) | GRM8GRM6GRM7GRM4GSR | |
| Glutamic Acid SCHEMBL2680237 | 0.86 | GRM8 (0.53) | GRM8GRM6GRM7GRM4GSR | |
| Glutamic Acid SCHEMBL9617054 | 0.85 | GRM8 (0.49) | GRM8GRM6GRM7GRM4GSR | |
| Glutamic Acid SCHEMBL9150210 | 0.85 | CYP1A2 (0.60) | GRM8GRM6GRM7GRM4GSR | |
| Aspartic Acid SCHEMBL15399013 | 0.82 | GRIK1 (0.38) | GRM8GRM6GRM7GRM4GSR | |
| Glycine SCHEMBL1548291 | 0.82 | SLC1A5 (0.38) | GRM8GRM6GRM7GRM4GSR | |
| SCHEMBL4752999 | 0.82 | SLC1A5 (0.40) | GRM8GRM6GRM7GRM4GSR |
Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.
Patent provenance — the patents this molecule appears in, and who filed them
Claimed or disclosed in 35 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.
| Patent | Title | Assignee | Published | Priority | Filing | Country | Status |
|---|---|---|---|---|---|---|---|
| EP-1137941-B1 | PROTEIN SCAFFOLDS FOR ANTIBODY MIMICS AND OTHER BINDING PROTEINS | BRISTOL MYERS SQUIBB CO (US) | 2009-08-12 | — | — | EP | claimed |
| EP-1137941-A4 | PROTEIN SCAFFOLDS FOR ANTIBODY MIMICS AND OTHER BINDING PROTEINS | PHYLOS INC (US) | 2002-04-17 | — | — | EP | claimed |
| EP-1137941-A1 | PROTEIN SCAFFOLDS FOR ANTIBODY MIMICS AND OTHER BINDING PROTEINS | Phylos, Inc. (US) | 2001-10-04 | — | — | EP | claimed |
| WO-2000034784-A9 | PROTEIN SCAFFOLDS FOR ANTIBODY MIMICS AND OTHER BINDING PROTEINS | PHYLOS INC (US) | 2000-11-16 | — | — | WO | claimed |
| WO-2000034784-A1 | PROTEIN SCAFFOLDS FOR ANTIBODY MIMICS AND OTHER BINDING PROTEINS | PHYLOS, INC. (US) | 2000-06-15 | — | — | WO | claimed |
| US-20170334958-A1 | PROTEIN SCAFFOLDS FOR ANTIBODY MIMICS AND OTHER BINDING PROTEINS | ADNEXUS, A BRISTOL-MYERS SQUIBB R&D COMPANY | 2017-11-23 | — | — | US | disclosed |
| US-20170275342-A1 | PROTEIN SCAFFOLDS FOR ANTIBODY MIMICS AND OTHER BINDING PROTEINS | BRISTOL MYERS SQUIBB CO (US) | 2017-09-28 | — | — | US | disclosed |
| US-9605039-B2 | Protein scaffolds for antibody mimics and other binding proteins | BRISTOL-MYERS SQUIBB COMPANY (US) | 2017-03-28 | — | — | US | disclosed |
| EP-1137941-B2 | PROTEIN SCAFFOLDS FOR ANTIBODY MIMICS AND OTHER BINDING PROTEINS | BRISTOL MYERS SQUIBB CO (US) | 2013-09-11 | — | — | EP | disclosed |
| EP-2154535-A1 | Protein scaffolds for antibody mimics and other binding proteins | Bristol-Myers Squibb Company (US) | 2010-02-17 | — | — | EP | disclosed |
| EP-2141243-A2 | Protein scaffolds for antibody mimics and other binding proteins | Brystol-Myers Squibb Company (US) | 2010-01-06 | — | — | EP | disclosed |
| EP-1137941-B1 | PROTEIN SCAFFOLDS FOR ANTIBODY MIMICS AND OTHER BINDING PROTEINS | BRISTOL MYERS SQUIBB CO (US) | 2009-08-12 | — | — | EP | disclosed |
| WO-2002032925-A9 | PROTEIN SCAFFOLDS FOR ANTIBODY MIMICS AND OTHER BINDING PROTEINS | PHYLOS INC (US) | 2003-02-06 | — | — | WO | disclosed |
| EP-1266025-A1 | PROTEIN SCAFFOLDS FOR ANTIBODY MIMICS AND OTHER BINDING PROTEINS | Compound Therapeutics, Inc. (US) | 2002-12-18 | — | — | EP | disclosed |
| WO-2002032925-A2 | PROTEIN SCAFFOLDS FOR ANTIBODY MIMICS AND OTHER BINDING PROTEINS | PHYLOS, INC. (US) | 2002-04-25 | — | — | WO | disclosed |
| EP-1137941-A4 | PROTEIN SCAFFOLDS FOR ANTIBODY MIMICS AND OTHER BINDING PROTEINS | PHYLOS INC (US) | 2002-04-17 | — | — | EP | disclosed |
| EP-1137941-A1 | PROTEIN SCAFFOLDS FOR ANTIBODY MIMICS AND OTHER BINDING PROTEINS | Phylos, Inc. (US) | 2001-10-04 | — | — | EP | disclosed |
| WO-2001064942-A1 | PROTEIN SCAFFOLDS FOR ANTIBODY MIMICS AND OTHER BINDING PROTEINS | PHYLOS, INC. (US) | 2001-09-07 | — | — | WO | disclosed |
| WO-2000034784-A9 | PROTEIN SCAFFOLDS FOR ANTIBODY MIMICS AND OTHER BINDING PROTEINS | PHYLOS INC (US) | 2000-11-16 | — | — | WO | disclosed |
| WO-2000034784-A1 | PROTEIN SCAFFOLDS FOR ANTIBODY MIMICS AND OTHER BINDING PROTEINS | PHYLOS, INC. (US) | 2000-06-15 | — | — | WO | disclosed |