SCHEMBL30724693

SCHEMBL30724693

CCOC(=O)c1cnc(NC2Cc3ccc(Br)cc3C2)cc1Cl

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.42
MAPT P10636 1/20 0.42
THRB P10828 1/20 0.42
MAPK1 P28482 1/20 0.42
RXFP1 Q9HBX9 3/20 0.41
NPSR1 Q6W5P4 1/20 0.41
OPRK1 P41145 2/20 0.40
PRMT5 O14744 1/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
NOS1 P29475 1/20 0.39
NOS2 P35228 1/20 0.39
DYRK1A Q13627 3/20 0.39
AURKA O14965 1/20 0.39
AURKB Q96GD4 1/20 0.39
ALDH1A1 P00352 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
JAK2 O60674 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27195418 1.00 GAA (0.42) GAAMAPTTHRBMAPK1RXFP1
SCHEMBL27195442 0.85 HDAC8 (0.40) MAPTOPRK1PRMT5NPC1RAB9A
SCHEMBL30724674 0.84 SORT1 (0.42) MAPTMAPK1PRMT5NPC1RAB9A
SCHEMBL27195343 0.84 SORT1 (0.42) MAPTMAPK1PRMT5NPC1RAB9A
SCHEMBL22092797 0.78 HDAC8 (0.43) GAAMAPK1RXFP1NPSR1OPRK1
SCHEMBL28653403 0.78 HDAC8 (0.43) GAAMAPK1RXFP1NPSR1OPRK1
SCHEMBL19190925 0.73 NNMT (0.61) MAPTNPC1RAB9AKMT2AALDH1A1
SCHEMBL27195353 0.72 HDAC8 (0.44) RXFP1PRMT5NPC1RAB9AMEN1
SCHEMBL30724696 0.72 HDAC8 (0.44) RXFP1PRMT5NPC1RAB9AMEN1
SCHEMBL4231706 0.72 P2RY12 (0.47) GAAMAPTNPC1RAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117396471-A Novel piperidine derivatives and pharmaceutical compositions for inhibiting autotaxin comprising the same 株式会社次代生物科学 2024-01-12 CN disclosed