SCHEMBL30740344

SCHEMBL30740344

Fc1cnn(-c2ccnc(Cl)n2)c1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 6/20 0.39
RPS6KA5 O75582 1/20 0.38
GRM5 P41594 2/20 0.38
TDO2 P48775 1/20 0.35
GABRA1 P14867 1/20 0.33
GABRG2 P18507 1/20 0.33
GABRB3 P28472 1/20 0.33
GABRA3 P34903 1/20 0.33
GRM4 Q14833 1/20 0.31
AR P10275 1/20 0.30
EGLN1 Q9GZT9 1/20 0.30
SORD Q00796 1/20 0.30
DYRK1B Q9Y463 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28606131 0.81 TRPV1 (0.43) TRPV1RPS6KA5GABRA1GABRG2GABRB3
SCHEMBL19100730 0.80 ALDH1A1 (0.41) TRPV1RPS6KA5TDO2
SCHEMBL31346256 0.80 TDO2 (0.35) GRM5TDO2GRM4DYRK1B
SCHEMBL18298616 0.80 RPS6KA5 (0.38) TRPV1RPS6KA5EGLN1SORD
SCHEMBL17670232 0.80 RPS6KA5 (0.35) TRPV1RPS6KA5EGLN1
SCHEMBL24920862 0.76 MAPT (0.34) GRM5TDO2GRM4EGLN1
SCHEMBL22071443 0.76 RPS6KA5 (0.35) TRPV1RPS6KA5
SCHEMBL31585397 0.76 GRM5 (0.39) RPS6KA5GRM5EGLN1
SCHEMBL19100794 0.76 RPS6KA5 (0.33) TRPV1RPS6KA5GABRA1GABRG2GABRB3
SCHEMBL24253886 0.75 GRM5 (0.39) GRM5TDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024022314-A1 TRIAZOLE COMPOUNDS AND USE THEREOF AS LPAR1 ANTAGONIST 武汉人福创新药物研发中心有限公司 2024-02-01 WO disclosed