SCHEMBL30744376

SCHEMBL30744376

N#Cc1cnn(Cc2ccc(C(F)(F)F)nc2)c1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 1/20 0.41
KCNH2 Q12809 1/20 0.39
GRIN1 Q05586 1/20 0.38
GRIN2B Q13224 1/20 0.38
CYP19A1 P11511 4/20 0.38
AR P10275 2/20 0.37
PGR P06401 1/20 0.37
RET P07949 1/20 0.37
CCR9 P51686 1/20 0.36
TRPV4 Q9HBA0 1/20 0.36
PDE9A O76083 2/20 0.36
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
GRM2 Q14416 1/20 0.35
P2RX3 P56373 1/20 0.35
P2RX2 Q9UBL9 1/20 0.35
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
DAO P14920 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21492003 1.00 KLKB1 (0.41) KLKB1KCNH2GRIN1GRIN2BCYP19A1
SCHEMBL17685589 0.82 KLKB1 (0.42) KLKB1CYP19A1ARPGRCYP11B1
SCHEMBL25269987 0.79 GRIN1 (0.40) KCNH2GRIN1GRIN2BRETTRPV4
SCHEMBL21503682 0.78 LOXL2 (0.40) KLKB1KCNH2GRIN1GRIN2BTRPV4
SCHEMBL21491519 0.77 GLS (0.38) KLKB1KCNH2GRIN1GRIN2BPGR
Hydrochloric Acid SCHEMBL21491894 0.77 LMNA (0.41) KLKB1KCNH2GRIN1GRIN2BTRPV4
SCHEMBL26202009 0.77 CYP3A4 (0.40) GRIN1GRIN2BTRPV4LMNAMAPT
Hydrochloric Acid SCHEMBL30744436 0.77 LMNA (0.41) KLKB1KCNH2GRIN1GRIN2BTRPV4
SCHEMBL24401098 0.76 GRIN1 (0.38) GRIN1GRIN2BTRPV4PDE9ACYP11B1
SCHEMBL21492571 0.76 GRIN1 (0.38) KCNH2GRIN1GRIN2BTRPV4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112218865-B Pteridinone compounds and uses thereof 沃泰克斯药物股份有限公司 2024-03-12 CN disclosed