SCHEMBL30745447

SCHEMBL30745447

COc1cc(O)c(C(=O)/C=C/c2ccc(F)cc2)cc1CNCc1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.60
BACE1 P56817 2/20 0.60
HDAC3 O15379 4/20 0.53
HDAC1 Q13547 4/20 0.53
HDAC2 Q92769 4/20 0.53
HDAC8 Q9BY41 4/20 0.53
CTSL P07711 2/20 0.52
APP P05067 2/20 0.52
TUBB4A P04350 1/20 0.50
TUBB P07437 1/20 0.50
TUBA3C P0DPH7 1/20 0.50
TUBA1B P68363 1/20 0.50
TUBA4A P68366 1/20 0.50
TUBB4B P68371 1/20 0.50
TUBB3 Q13509 1/20 0.50
TUBB2A Q13885 1/20 0.50
TUBB8 Q3ZCM7 1/20 0.50
TUBA3E Q6PEY2 1/20 0.50
TUBA1A Q71U36 1/20 0.50
TUBA1C Q9BQE3 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30745479 0.91 APP (0.52) ACHEBACE1HDAC3HDAC1HDAC2
SCHEMBL30745475 0.90 ABCG2 (0.52) ACHEBACE1HDAC3HDAC1HDAC2
SCHEMBL30745466 0.89 MAOA (0.53) HDAC3HDAC1HDAC2HDAC8APP
SCHEMBL30745477 0.81 HDAC3 (0.55) ACHEBACE1HDAC3HDAC1HDAC2
SCHEMBL25239854 0.79 ACHE (0.81) ACHEBACE1CTSLTUBB4ATUBB
SCHEMBL30745430 0.79 ACHE (0.67) ACHEBACE1CTSLTUBB4ATUBB
SCHEMBL30745488 0.79 ACHE (0.65) ACHEBACE1CTSLAPPTUBB4A
SCHEMBL29011908 0.76 ACHE (0.76) ACHEBACE1CTSLAPPTUBB4A
SCHEMBL30745514 0.75 ACHE (0.61) ACHEBACE1CTSLAPPMAOB
SCHEMBL30745510 0.75 ABCG2 (0.53) ACHEBACE1ARMAOBABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117567303-A Chalcone Mannich base compound, pharmaceutical composition, preparation method and application thereof 安徽中医药大学 2024-02-20 CN claimed
CN-117567303-A Chalcone Mannich base compound, pharmaceutical composition, preparation method and application thereof 安徽中医药大学 2024-02-20 CN disclosed