SCHEMBL30760160

SCHEMBL30760160

Cc1cnccc1-c1ccc([C@H](CO)NC(=O)C2CCCN2O)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 5/20 0.46
ABL1 P00519 1/20 0.39
ROCK2 O75116 6/20 0.39
ROCK1 Q13464 3/20 0.39
CCR5 P51681 1/20 0.38
KCNH2 Q12809 1/20 0.38
RPS6KA5 O75582 2/20 0.37
MAP4K4 O95819 2/20 0.37
PRKCG P05129 2/20 0.37
CDK1 P06493 2/20 0.37
PRKACA P17612 2/20 0.37
RPS6KB1 P23443 2/20 0.37
CDK2 P24941 2/20 0.37
AKT1 P31749 2/20 0.37
AKT2 P31751 2/20 0.37
CLK2 P49760 2/20 0.37
GSK3A P49840 2/20 0.37
GSK3B P49841 2/20 0.37
IRAK1 P51617 2/20 0.37
RPS6KA3 P51812 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30760076 0.78 MAPK1 (0.60) MAPK1ROCK2ROCK1RPS6KA5MAP4K4
SCHEMBL27360361 0.78 MAPK1 (0.38) MAPK1
SCHEMBL30760039 0.77 MAPK1 (0.46) MAPK1ABL1ROCK2ROCK1RPS6KA5
SCHEMBL30760172 0.74 CYP1A2 (0.47) MAPK1CYP3A4
SCHEMBL30760038 0.74 VHL (0.51) MAPK1
SCHEMBL3104408 0.73 MAPK1 (0.67) MAPK1ROCK2ROCK1RPS6KA5MAP4K4
SCHEMBL27360587 0.72 PTGES (0.35) MAPK1ABL1CCR5KCNH2BRAF
SCHEMBL30760184 0.72 MAPK1 (0.51) MAPK1ROCK2ROCK1RPS6KA5MAP4K4
SCHEMBL27360367 0.71 XIAP (0.38) ABL1PTGESPTGS2
SCHEMBL27360586 0.71 DPP4 (0.40) MAPK1ABL1CCR5KCNH2BRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024040080-A1 KRAS INHIBITOR CONJUGATES ERASCA, INC. (US) 2024-02-22 WO disclosed