SCHEMBL30780893

SCHEMBL30780893

Nc1ccn(-c2cc(C(F)(F)F)cc(C(F)(F)F)c2)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
AR P10275 1/20 0.40
NOS3 P29474 1/20 0.39
NOS2 P35228 1/20 0.39
NOTUM Q6P988 3/20 0.38
ADRB1 P08588 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
NR2E1 Q9Y466 1/20 0.36
ALOX5 P09917 1/20 0.36
PTGS1 P23219 1/20 0.36
PTGS2 P35354 1/20 0.36
CASR P41180 2/20 0.35
PKM P14618 1/20 0.35
BACE1 P56817 1/20 0.35
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
EPHX2 P34913 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL45043 0.85 NOTUM (0.56) ALDH1A1NOTUMCYP1A2CYP3A4CYP2C9
SCHEMBL11614453 0.84 CASR (0.46) ALDH1A1NOTUMPTGS2CASR
Hydrochloric Acid SCHEMBL1082574 0.83 NOTUM (0.55) ALDH1A1NOTUMCYP1A2CYP3A4CYP2C9
SCHEMBL19281408 0.79 AR (0.43) ALDH1A1ARNOTUMADRB1CYP1A2
SCHEMBL28223159 0.78 GABRA2 (0.47)
SCHEMBL16056137 0.76 NR2E1 (0.54) ALDH1A1ARNOTUMCYP1A2CYP3A4
SCHEMBL380712 0.76 L3MBTL1 (0.40) ALDH1A1CYP3A4BACE1
SCHEMBL4868706 0.73 AR (0.45) ARNOTUM
SCHEMBL20242016 0.73 AR (0.43) ARNOS3NOS2NOTUM
SCHEMBL31052478 0.71 DHFR (0.44) CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024030651-A1 GPX4 INHIBITORS AND USE THEREOF SONATA THERAPEUTICS, INC. (US) 2024-02-08 WO disclosed