SCHEMBL20242016

SCHEMBL20242016

Nc1ccn(-c2ccnc(C(F)(F)F)c2)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.43
LOXL2 Q9Y4K0 2/20 0.42
LOX P28300 1/20 0.41
GRIN1 Q05586 3/20 0.40
GRIN2B Q13224 3/20 0.40
RXRA P19793 2/20 0.40
CA2 P00918 1/20 0.40
CHKA P35790 1/20 0.40
NOS3 P29474 1/20 0.39
NOS2 P35228 1/20 0.39
CYP17A1 P05093 1/20 0.37
IDH1 O75874 3/20 0.35
PRMT6 Q96LA8 1/20 0.35
KDM4E B2RXH2 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MAP4K4 O95819 1/20 0.35
NOTUM Q6P988 1/20 0.34
IDO1 P14902 1/20 0.34
ELOVL1 Q9BW60 1/20 0.34
PARP1 P09874 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15825104 0.84 AR (0.43) ARLOXL2LOXGRIN1GRIN2B
SCHEMBL28393138 0.81 NOS3 (0.46) LOXL2CA2CHKANOS3NOS2
SCHEMBL15832232 0.81 AR (0.46) ARLOXL2LOXGRIN1GRIN2B
SCHEMBL20241939 0.80 ELOVL1 (0.43) NOS3NOS2KDM4EELOVL1
SCHEMBL20241993 0.79 ELOVL1 (0.42) LOXL2NOS3NOS2L3MBTL1MAP4K4
SCHEMBL17356153 0.78 AR (0.43) ARLOXL2LOXGRIN1GRIN2B
SCHEMBL31052478 0.76 DHFR (0.44) CA2CHKAIDH1PRMT6MAP4K4
SCHEMBL20242276 0.76 ELOVL1 (0.40) GRIN1GRIN2BRXRANOS3NOS2
SCHEMBL20242055 0.76 LOX (0.38) LOXL2LOXCYP17A1NOTUMELOVL1
SCHEMBL20241821 0.76 ELOVL1 (0.36) NOS3NOS2ELOVL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180251431-A1 1,3-SUBSTITUTED PYRAZOLE COMPOUNDS USEFUL FOR REDUCTION OF VERY LONG CHAIN FATTY ACID LEVELS VERTEX PHARMACEUTICALS INCORPORATED 2018-09-06 US disclosed
WO-2018107056-A1 1,3-SUBSTITUED PYRAZOLE COMPOUNDS USEFUL FOR REDUCTION OF VERY LONG CHAIN FATTY ACIC LEVELS VERTEX PHARMACEUTICALS INCORPORATED (US) 2018-06-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180251431-A1 1,3-SUBSTITUTED PYRAZOLE COMPOUNDS USEFUL FOR REDUCTION OF VERY LONG CHAIN FATTY ACID LEVELS HSD17B4, CPT1A, ADH1A AR 707/4885LOXL2 2328/4885LOX 2604/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.