SCHEMBL307974

SCHEMBL307974

NC(=O)C1(C(N)=O)CC1c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 16/20 0.48
MAOA P21397 16/20 0.48
MAOB P27338 16/20 0.48
MAPK1 P28482 1/20 0.44
CYP2C19 P33261 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2401865 0.92 KDM1A (0.46) KDM1AMAOAMAOBMAPK1CYP2C19
SCHEMBL28206522 0.89 KDM1A (0.43) KDM1AMAOAMAOBMAPK1CYP2C19
SCHEMBL5435422 0.83 MAPK1 (0.50) KDM1AMAOAMAOBMAPK1CYP2C19
SCHEMBL28521164 0.81 KDM1A (0.45) KDM1AMAOAMAOBMAPK1
SCHEMBL28511550 0.81 KDM1A (0.45) KDM1AMAOAMAOB
SCHEMBL28519822 0.81 ALDH1A1 (0.40) MAOAMAOBCYP2C19
SCHEMBL900614 0.81 KDM1A (0.45) KDM1AMAOAMAOB
SCHEMBL28524795 0.80 KDM1A (0.51) KDM1A
SCHEMBL9452686 0.80 KDM1A (0.39) KDM1AMAOAMAOB
Hydrochloric Acid SCHEMBL29430083 0.79 KDM1A (0.47) KDM1AMAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8093264-B2 Fused heterocycles as inhibitors of VEGF receptor and HGF receptor signaling METHYLGENE INC. (CA) 2012-01-10 US claimed
US-20070004675-A1 Inhibitors of VEGF receptor and HGF receptor signaling METHYLGENE, INC. 2007-01-04 US claimed
EP-1377589-A1 OXAZOLYL-PYRAZOLE DERIVATIVES AS KINASE INHIBITORS Pharmacia Italia S.p.A. (IT) 2004-01-07 EP claimed
WO-2002062804-A1 OXAZOLYL-PYRAZOLE DERIVATIVES AS KINASE INHIBITORS PHARMACIA ITALIA S.P.A. (IT) 2002-08-15 WO claimed
CN-112142619-B 1, 1-cyclopropane dicarboxylic acid amide compound and preparation method and application thereof 浙江工业大学 2023-01-10 CN disclosed
CN-112142619-A 1, 1-cyclopropane dicarboxylic acid amide compound and preparation method and application thereof 浙江工业大学 2020-12-29 CN disclosed
WO-2010045095-A1 COMPOUNDS AND METHODS OF USE XI NING (US) 2010-04-22 WO disclosed
WO-2009136663-A1 FUSED HETEROCYCLIC DERIVATIVES AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070004675-A1 Inhibitors of VEGF receptor and HGF receptor signaling HGF, MET, FLT1 KDM1A 4241/4885MAOA 3677/4885MAOB 3560/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.