SCHEMBL30823972

SCHEMBL30823972

NC(=O)c1ncc2n1CCOC2

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.35
HTT P42858 1/20 0.35
POLB P06746 1/20 0.34
JAK2 O60674 2/20 0.32
JAK1 P23458 2/20 0.32
TYK2 P29597 2/20 0.32
JAK3 P52333 2/20 0.32
CYP11B2 P19099 1/20 0.32
AURKA O14965 1/20 0.32
RPS6KB1 P23443 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
F10 P00742 1/20 0.31
ALDH1A1 P00352 1/20 0.31
PIK3CA P42336 1/20 0.30
MTOR P42345 1/20 0.30
HPGD P15428 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25333075 0.73 SSTR4 (0.40) KDM4EHTTALDH1A1HPGD
SCHEMBL15432302 0.71 TGFBR1 (0.37)
SCHEMBL16906805 0.71 TGFBR1 (0.37) KDM4EALDH1A1HPGD
SCHEMBL24729111 0.71 CA12 (0.34) POLBALDH1A1
SCHEMBL19659000 0.71 RIPK1 (0.47)
SCHEMBL24729109 0.70 ALDH1A1 (0.32) ALDH1A1
SCHEMBL12408124 0.70 SMN1; SMN2 (0.32) KDM4EHTTSMN1; SMN2ALDH1A1PIK3CA
SCHEMBL15451930 0.68 PARP2 (0.41) KDM4ESMN1; SMN2ALDH1A1HPGD
SCHEMBL24729110 0.68 ALDH1A1 (0.31) POLBALDH1A1
SCHEMBL24729048 0.68

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3760625-B1 BICYCLIC LACTAMS AS RECEPTOR-INTERACTING PROTEIN-1 (RIP1) KINASE INHIBITORS FOR TREATING E.G. INFLAMMATORY DISEASES HOFFMANN LA ROCHE (CH) 2024-03-27 EP claimed