SCHEMBL30832005

SCHEMBL30832005

COCc1ccc(CNC(=O)NCC2CCN(CC(=O)c3ccc(F)cc3)CC2)cc1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.48
MEN1 O00255 1/20 0.48
CCR3 P51677 1/20 0.46
MCHR1 Q99705 1/20 0.43
ALDH1A1 P00352 1/20 0.42
POLB P06746 1/20 0.42
GAA P10253 1/20 0.42
LMNA P02545 1/20 0.42
TSHR P16473 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
KCNH2 Q12809 2/20 0.42
CACNA1I Q9P0X4 1/20 0.42
HTR2A P28223 2/20 0.42
HTR2C P28335 1/20 0.42
HTR1A P08908 1/20 0.42
TMEM97 Q5BJF2 1/20 0.42
HTR4 Q13639 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL29207934 0.95 KMT2A (0.45) KMT2AMEN1CCR3ALDH1A1POLB
SCHEMBL30832018 0.88 KMT2A (0.43) KMT2AMEN1CCR3ALDH1A1POLB
SCHEMBL30831997 0.85 HTR2A (0.48) KMT2AMEN1ALDH1A1GAATSHR
SCHEMBL30832012 0.85 HTR2A (0.46) KMT2ALMNATSHRSMN1; SMN2KCNH2
Trifluoroacetic Acid SCHEMBL29208021 0.84 KMT2A (0.40) KMT2AMEN1CCR3ALDH1A1POLB
SCHEMBL30831994 0.84 KMT2A (0.42) KMT2AMEN1ALDH1A1POLBGAA
SCHEMBL29207983 0.82 HTR2A (0.49) KMT2AKCNH2HTR2AHTR2C
Trifluoroacetic Acid SCHEMBL29280883 0.82 SMN1; SMN2 (0.48) KMT2APOLBLMNATSHRSMN1; SMN2
SCHEMBL30834063 0.82 LMNA (0.46) KMT2AMEN1ALDH1A1GAALMNA
SCHEMBL30832034 0.82 HRH3 (0.51) LMNATSHRSMN1; SMN2KCNH2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117964547-A Urea compound and application thereof as Sigma2 and 5HT2A dual-target inhibitor 瀚远医药有限公司 2024-05-03 CN disclosed
WO-2024067304-A1 COMPOUND WITH INHIBITORY ACTIVITY AGAINST SIGMA2 AND 5HT2A AND USE 瀚远医药有限公司 2024-04-04 WO disclosed