SCHEMBL30832010

SCHEMBL30832010

COc1ccc(CN(C)C(=O)NCC2CCN(CC(=O)c3ccc(F)cc3)CC2)cn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
HTR4 Q13639 1/20 0.40
KDM1A O60341 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
ALDH1A1 P00352 2/20 0.38
POLB P06746 1/20 0.38
GAA P10253 1/20 0.38
F10 P00742 2/20 0.38
GRIN2B Q13224 1/20 0.38
GSK3B P49841 2/20 0.38
KDM4E B2RXH2 1/20 0.38
TSHR P16473 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HTR1A P08908 1/20 0.38
HTR2A P28223 1/20 0.38
TMEM97 Q5BJF2 1/20 0.38
ATM Q13315 1/20 0.38
PRKAB2 O43741 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL29208031 0.95 GSK3B (0.38) MEN1KMT2AHTR4KDM1AHDAC6
SCHEMBL30842029 0.88 HTR4 (0.39) MEN1KMT2AHTR4ALDH1A1POLB
SCHEMBL30832023 0.87 MLLT1 (0.43) ALDH1A1GRIN2BKDM4ETSHRHTT
SCHEMBL30831994 0.85 KMT2A (0.42) MEN1KMT2AHTR4ALDH1A1POLB
Trifluoroacetic Acid SCHEMBL29207962 0.84 HTR2A (0.38) MEN1KMT2AHTR4HTR2A
Trifluoroacetic Acid SCHEMBL29207943 0.83 MLLT1 (0.40) GRIN2BHTR2APRKAB2PRKAG1PRKAA2
SCHEMBL30832017 0.81 SMN1; SMN2 (0.42) MEN1KMT2AALDH1A1KDM4ETSHR
Trifluoroacetic Acid SCHEMBL29208017 0.81 CHRM4 (0.40) MEN1KMT2AHTR4HTR1AHTR2A
SCHEMBL30832020 0.80 ALDH1A1 (0.42) MEN1KMT2AKDM1AHDAC6ALDH1A1
Trifluoroacetic Acid SCHEMBL29280867 0.79 GABRA5 (0.48) KDM1AHDAC6F10GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117964547-A Urea compound and application thereof as Sigma2 and 5HT2A dual-target inhibitor 瀚远医药有限公司 2024-05-03 CN disclosed
WO-2024067304-A1 COMPOUND WITH INHIBITORY ACTIVITY AGAINST SIGMA2 AND 5HT2A AND USE 瀚远医药有限公司 2024-04-04 WO disclosed