SCHEMBL30833699

SCHEMBL30833699

O=[SH](=O)NCc1ccccc1Nc1nc(Nc2ccc3c(N4CCOCC4)n[nH]c3c2)ncc1Cl

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 3/20 0.49
CCNK O75909 1/20 0.49
CCNA2 P20248 1/20 0.49
CDK2 P24941 1/20 0.49
CCND3 P30281 1/20 0.49
CDK9 P50750 1/20 0.49
CDK6 Q00534 1/20 0.49
ALK Q9UM73 4/20 0.49
PKMYT1 Q99640 2/20 0.49
AXL P30530 1/20 0.49
INSR P06213 1/20 0.49
IGF1R P08069 1/20 0.49
PTK2 Q05397 1/20 0.49
PTK2B Q14289 1/20 0.49
SLC2A1 P11166 1/20 0.48
MAPK9 P45984 4/20 0.48
MAPK10 P53779 4/20 0.48
MAPK8 P45983 2/20 0.48
ULK1 O75385 1/20 0.47
MAP3K7 O43318 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30833672 0.87 ALK (0.51) EGFRCCNKCCNA2CDK2CCND3
SCHEMBL30833785 0.85 ALK (0.51) EGFRALKIGF1RMAPK9MAPK10
SCHEMBL29190631 0.85 IGF1R (0.44) EGFRALKIGF1RPTK2
SCHEMBL30833687 0.84 ALK (0.50) EGFRALKMAPK9MAPK10ULK1
SCHEMBL29190617 0.84 ALK (0.68) EGFRCCNKCCNA2CDK2CCND3
SCHEMBL29190716 0.83 FGFR1 (0.44) EGFRCDK2ALKIGF1RPTK2
SCHEMBL30833656 0.83 ALK (0.48) ALKAXLIGF1R
SCHEMBL30833633 0.81 EGFR (0.47) EGFRCDK2ALKPTK2PTK2B
SCHEMBL30833661 0.79 ALK (0.46) CCNKCCNA2CDK2CCND3CDK9
SCHEMBL30833669 0.77 ALK (0.46) CCNKCCNA2CDK2CCND3CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113896744-B Selective EGFR inhibitor 成都先导药物开发股份有限公司 2024-04-16 CN disclosed