SCHEMBL30833644

SCHEMBL30833644

O=[N+]([O-])c1ccc2c(N3CC(CO)C3)n[nH]c2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.43
DAO P14920 1/20 0.42
PNMT P11086 2/20 0.41
ADRA2A P08913 1/20 0.41
MAPT P10636 2/20 0.40
HPGD P15428 1/20 0.40
MAP2K7 O14733 1/20 0.39
CYP3A4 P08684 2/20 0.38
LMNA P02545 1/20 0.38
ALOX15 P16050 1/20 0.38
NOS1 P29475 1/20 0.38
GSK3B P49841 2/20 0.38
PARP1 P09874 1/20 0.37
CDK2 P24941 1/20 0.37
PKM P14618 2/20 0.37
GBA1 P04062 1/20 0.36
NAMPT P43490 1/20 0.36
XDH P47989 1/20 0.36
CYP1A2 P05177 1/20 0.36
PKLR P30613 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29190572 1.00 MAPK1 (0.43) MAPK1DAOPNMTADRA2AMAPT
SCHEMBL30833670 0.83 HTT (0.54) DAOPNMTADRA2AMAPTHPGD
SCHEMBL30833712 0.78 MAPK1 (0.44) MAPK1GSK3B
SCHEMBL29190564 0.78 MAPK1 (0.44) MAPK1GSK3B
SCHEMBL30833685 0.78 MAPK1 (0.52) MAPK1MAPTHPGDLMNACYP1A2
SCHEMBL29190669 0.78 MAPK1 (0.52) MAPK1MAPTHPGDLMNACYP1A2
SCHEMBL30833799 0.78 SIRT6 (0.50) MAPK1MAPTHPGDCYP3A4LMNA
SCHEMBL4784574 0.78 SIRT6 (0.50) MAPK1MAPTHPGDCYP3A4LMNA
SCHEMBL1489156 0.73 MAPT (0.47) DAOMAPTHPGDMAP2K7CYP3A4
SCHEMBL22445861 0.71 MAPT (0.47) MAPTHPGDLMNACDK2PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113896744-B Selective EGFR inhibitor 成都先导药物开发股份有限公司 2024-04-16 CN disclosed