SCHEMBL30833786

SCHEMBL30833786

NS(=O)(=O)Cc1ccccc1Nc1nc(Nc2ccc3nccnc3c2)ncc1Br

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.48
MAPK8 P45983 3/20 0.44
SYK P43405 3/20 0.44
IGF1R P08069 5/20 0.44
CDK1 P06493 4/20 0.44
CDK2 P24941 3/20 0.44
KDR P35968 3/20 0.44
ALK Q9UM73 2/20 0.44
GSK3B P49841 2/20 0.44
PTK2 Q05397 2/20 0.44
AURKA O14965 2/20 0.44
AURKB Q96GD4 2/20 0.44
CDC7 O00311 1/20 0.44
PLK4 O00444 1/20 0.44
CHEK1 O14757 1/20 0.44
DCLK1 O15075 1/20 0.44
MAPK13 O15264 1/20 0.44
PDPK1 O15530 1/20 0.44
DAPK3 O43293 1/20 0.44
DYRK3 O43781 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30833742 0.85 IGF1R (0.43) EGFRMAPK8SYKIGF1RCDK1
SCHEMBL30833774 0.85 IGF1R (0.43) MAPK8SYKIGF1RCDK1CDK2
SCHEMBL30833734 0.84 ALK (0.49) EGFRMAPK8SYKIGF1RCDK1
SCHEMBL30833779 0.83 EGFR (0.48) EGFRMAPK8SYKIGF1RCDK1
SCHEMBL30833668 0.83 EGFR (0.52) EGFRALKJAK2FGFR1SRC
SCHEMBL30833660 0.82 ALK (0.43) EGFRMAPK8SYKIGF1RCDK1
SCHEMBL29190693 0.81 GLO1 (0.54) EGFRMAPK8IGF1RCDK1CDK2
SCHEMBL30833764 0.79 IGF1R (0.45) EGFRMAPK8SYKIGF1RCDK1
SCHEMBL30833715 0.78 SYK (0.46) MAPK8SYKIGF1RCDK1CDK2
SCHEMBL30833796 0.76 IGF1R (0.46) EGFRMAPK8IGF1RCDK1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113896744-B Selective EGFR inhibitor 成都先导药物开发股份有限公司 2024-04-16 CN disclosed