SCHEMBL30833869

SCHEMBL30833869

C#Cc1ccc(-c2nnc(NC3CCCNC3)cc2C(F)(F)F)c(O)c1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
IL1B P01584 10/20 0.51
NLRP3 Q96P20 6/20 0.51
CCNK O75909 6/20 0.42
CDK12 Q9NYV4 6/20 0.42
CDK7 P50613 4/20 0.42
CCNH P51946 4/20 0.42
CCNT1 O60563 4/20 0.42
CCNE1 P24864 4/20 0.42
CDK2 P24941 4/20 0.42
CDK9 P50750 4/20 0.42
MNAT1 P51948 3/20 0.42
PIM1 P11309 1/20 0.40
TNF P01375 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30834025 1.00 IL1B (0.51) IL1BNLRP3CCNKCDK12CDK7
SCHEMBL30833946 0.85 NLRP3 (0.55) IL1BNLRP3TNF
SCHEMBL25302079 0.85 NLRP3 (0.42) IL1BNLRP3CCNKCDK12CDK7
SCHEMBL30488537 0.85 NLRP3 (0.42) IL1BNLRP3CCNKCDK12CDK7
SCHEMBL25262878 0.85 NLRP3 (0.42) IL1BNLRP3CCNKCDK12CDK7
SCHEMBL30488601 0.85 NLRP3 (0.42) IL1BNLRP3CCNKCDK12CDK7
SCHEMBL30833973 0.81 IL1B (0.77) IL1BNLRP3
SCHEMBL30833859 0.80 IL1B (0.74) IL1BNLRP3TNF
SCHEMBL31681934 0.79 IL1B (0.59) IL1BNLRP3TNF
SCHEMBL30833951 0.79 IL1B (0.59) IL1BNLRP3TNF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117986258-A NLRP3 inflammation corpuscle inhibitor and application thereof 药捷安康(南京)科技股份有限公司 2024-05-07 CN disclosed