SCHEMBL30844573

SCHEMBL30844573

Cc1onc(NS(=O)(=O)c2ccccc2Br)c1Cl

nearest known ligand 0.56

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 11/20 0.56
EDNRB P24530 9/20 0.56
BRD4 O60885 1/20 0.49
FBP1 P09467 1/20 0.44
ALDH1A1 P00352 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5330400 1.00 EDNRA (0.56) EDNRAEDNRBBRD4FBP1ALDH1A1
SCHEMBL30171185 0.86 EDNRA (0.63) EDNRAEDNRBBRD4
SCHEMBL5529599 0.86 EDNRA (0.63) EDNRAEDNRBBRD4
SCHEMBL30296336 0.84 EDNRA (0.56) EDNRAEDNRBBRD4FBP1
SCHEMBL5321684 0.84 EDNRA (0.56) EDNRAEDNRBBRD4FBP1
SCHEMBL29281015 0.83 EDNRA (0.45) EDNRAEDNRB
SCHEMBL30296058 0.82 EDNRA (0.66) EDNRAEDNRBFBP1
SCHEMBL7222597 0.80 EDNRB (0.61) EDNRAEDNRBBRD4ALDH1A1RXFP1
SCHEMBL9063934 0.80 EDNRB (0.61) EDNRAEDNRBBRD4ALDH1A1RXFP1
SCHEMBL24822840 0.80 EDNRA (0.43) EDNRAEDNRBALDH1A1RXFP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250051315-A1 COMPOUND, ANGIOTENSIN II TYPE 1 RECEPTOR ANTAGONIST AND PHARMACEUTICAL COMPOSITION ALCHEMEDICINE, INC. (JP) 2025-02-13 US disclosed
EP-4458826-A1 COMPOUND, ANGIOTENSIN II TYPE 1 RECEPTOR ANTAGONIST AND PHARMACEUTICAL COMPOSITION Alchemedicine, Inc. (JP) 2024-11-06 EP disclosed
CN-118546134-A Crystal form containing aromatic ring derivative antagonist, preparation method and application thereof 江苏豪森药业集团有限公司 2024-08-27 CN disclosed
CN-118284605-A Compounds, angiotensin II type 1 receptor antagonists and pharmaceutical compositions 亚克医药株式会社 2024-07-02 CN disclosed
CN-117836294-A Biological antagonist containing aromatic ring, preparation method and application thereof 上海翰森生物医药科技有限公司 2024-04-05 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250051315-A1 COMPOUND, ANGIOTENSIN II TYPE 1 RECEPTOR ANTAGONIST AND PHARMACEUTICAL COMPOSITION AGTR1, AGTR2, ADRB1 EDNRA 154/4885EDNRB 216/4885BRD4 915/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.