SCHEMBL30850107

SCHEMBL30850107

COC(=O)C1=CN=C2N=CN=C2C1

nearest known ligand 0.33

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 2/20 0.33
LMNA P02545 1/20 0.32
CHRM2 P08172 1/20 0.32
CHRM4 P08173 1/20 0.32
CHRM5 P08912 1/20 0.32
THRB P10828 1/20 0.32
CHRM1 P11229 1/20 0.32
BLM P54132 1/20 0.31
MCOLN3 Q8TDD5 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
MAPK1 P28482 1/20 0.30
CA12 O43570 1/20 0.30
CA9 Q16790 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1759161 0.80
SCHEMBL29053129 0.74 CA12 (0.33) CHRM3LMNACHRM2CHRM4CHRM5
SCHEMBL1895595 0.73 CHRM3 (0.32) CHRM3LMNACHRM2CHRM4CHRM5
SCHEMBL30051946 0.71 CHRM3 (0.33) CHRM3LMNACHRM2CHRM4CHRM5
SCHEMBL30731288 0.69 CA12 (0.32) CHRM3LMNACHRM2CHRM4CHRM5
SCHEMBL3664888 0.68 CA12 (0.35) CHRM3LMNACHRM2CHRM4CHRM5
SCHEMBL1870026 0.68 TRPA1 (0.31) NPSR1
SCHEMBL18104379 0.65 MAPK1 (0.41) MAPK1
SCHEMBL23280497 0.63 CHRM3 (0.37) CHRM3LMNACHRM2CHRM4CHRM5
SCHEMBL21277825 0.60 LOXL2 (0.40) CHRM3LMNACHRM2CHRM4CHRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115551862-B Macrocyclic inhibitors of peptidyl arginine deiminase 吉利德科学公司 2024-04-12 CN disclosed