SCHEMBL30857596

SCHEMBL30857596

COC(=O)c1ccc2c(c1)N(CCO[Si](C)(C)C(C)(C)C)C[C@@H]1CN(CC3=C(c4ccc(Cl)cc4)CCC(C)(C)C3)CCN21

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
BCL2L1 Q07817 14/20 0.44
BCL2 P10415 17/20 0.42
BCL2L11 O43521 1/20 0.36
CYP2C9 P11712 1/20 0.36
MCL1 Q07820 1/20 0.36
ASPH Q12797 1/20 0.36
BCL2L2 Q92843 1/20 0.36
BAD Q92934 1/20 0.36
USP2 O75604 1/20 0.35
ALOX15 P16050 1/20 0.35
HSD17B10 Q99714 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30857714 0.81 BCL2L1 (0.57) BCL2L1BCL2BCL2L11CYP2C9MCL1
SCHEMBL30857713 0.80 BCL2L1 (0.50) BCL2L1BCL2BCL2L11CYP2C9MCL1
SCHEMBL30857518 0.80 BCL2L1 (0.50) BCL2L1BCL2BCL2L11CYP2C9MCL1
SCHEMBL30857664 0.75 BCL2L1 (0.50) BCL2L1BCL2USP2ALOX15HSD17B10
SCHEMBL30857621 0.73 BCL2L1 (0.41) BCL2L1BCL2USP2ALOX15HSD17B10
SCHEMBL21751667 0.73 BCL2L1 (0.59) BCL2L1BCL2BCL2L11CYP2C9MCL1
SCHEMBL30857549 0.73 BCL2L1 (0.50) BCL2L1BCL2BCL2L11CYP2C9MCL1
SCHEMBL5128722 0.72 BCL2L1 (0.61) BCL2L1BCL2BAD
SCHEMBL5128718 0.72 BCL2L1 (0.61) BCL2L1BCL2BAD
SCHEMBL30857660 0.72 BCL2L1 (0.58) BCL2L1BCL2BCL2L11CYP2C9MCL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024067818-A1 CHIMERIC COMPOUND USED FOR TARGETED DEGRADATION OF BCL-2 PROTEIN, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL APPLICATION THEREOF 江苏恒瑞医药股份有限公司 2024-04-04 WO disclosed