SCHEMBL30865616

SCHEMBL30865616

CC(C)c1cnc(C(=O)N[C@H]2C[C@H](O)C2)c2cnc(Cl)cc12

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 3/20 0.39
ADORA2A P29274 2/20 0.39
CNR2 P34972 9/20 0.37
HPGDS O60760 1/20 0.37
CHRM5 P08912 1/20 0.36
BRD4 O60885 1/20 0.36
TRPV1 Q8NER1 2/20 0.35
ADORA1 P30542 1/20 0.35
MAP4K4 O95819 1/20 0.34
RORC P51449 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24813085 1.00 ADORA2B (0.39) ADORA2BADORA2ACNR2HPGDSCHRM5
SCHEMBL24811658 0.86 CNR2 (0.35) CNR2BRD4
SCHEMBL30865622 0.86 CNR2 (0.35) CNR2BRD4
SCHEMBL29239449 0.85 HPGDS (0.41) CNR2HPGDS
SCHEMBL24811744 0.85 HPGDS (0.41) CNR2HPGDS
SCHEMBL30865627 0.85 CNR2 (0.48) CNR2HPGDSBRD4TRPV1
SCHEMBL24811650 0.85 CNR2 (0.48) CNR2HPGDSBRD4TRPV1
SCHEMBL24810635 0.85 IRAK4 (0.35) CNR2TRPV1
SCHEMBL30164503 0.85 IRAK4 (0.35) CNR2TRPV1
SCHEMBL24810238 0.82 HTR4 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117916232-A Heterocyclic EGFR inhibitors for the treatment of cancer 缆图药品公司 2024-04-19 CN disclosed