SCHEMBL30865627

SCHEMBL30865627

CC(C)c1cnc(C(=O)NC2CCOCC2)c2cnc(Cl)cc12

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 9/20 0.48
TRPV1 Q8NER1 2/20 0.41
HTR4 Q13639 2/20 0.39
HPGDS O60760 1/20 0.39
PTGER1 P34995 1/20 0.38
BRD4 O60885 2/20 0.38
DYRK1A Q13627 1/20 0.38
NPC1 O15118 1/20 0.37
TSHR P16473 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
SELP P16109 1/20 0.36
TYRO3 Q06418 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24811650 1.00 CNR2 (0.48) CNR2TRPV1HTR4HPGDSPTGER1
SCHEMBL24813085 0.85 ADORA2B (0.39) CNR2TRPV1HPGDSBRD4
SCHEMBL30865616 0.85 ADORA2B (0.39) CNR2TRPV1HPGDSBRD4
SCHEMBL29239449 0.82 HPGDS (0.41) CNR2HPGDS
SCHEMBL24811744 0.82 HPGDS (0.41) CNR2HPGDS
SCHEMBL24811658 0.81 CNR2 (0.35) CNR2BRD4
SCHEMBL30865622 0.81 CNR2 (0.35) CNR2BRD4
SCHEMBL24810635 0.80 IRAK4 (0.35) CNR2TRPV1DYRK1A
SCHEMBL30164503 0.80 IRAK4 (0.35) CNR2TRPV1DYRK1A
SCHEMBL24810238 0.79 HTR4 (0.39) HTR4DYRK1ACYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117916232-A Heterocyclic EGFR inhibitors for the treatment of cancer 缆图药品公司 2024-04-19 CN disclosed