SCHEMBL30872154

SCHEMBL30872154

Cc1cc(C)nc(-n2cc3c(c2)CN(C(=O)c2c(-c4ccccc4)nn4ccncc24)C3)n1

nearest known ligand 0.37

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 13/20 0.37
HCRTR1 O43613 12/20 0.37
EGFR P00533 1/20 0.35
HSP90AA1 P07900 1/20 0.34
SLC6A7 Q99884 1/20 0.33
ALDH1A1 P00352 2/20 0.33
HTT P42858 1/20 0.33
USP2 O75604 1/20 0.33
KDM4E B2RXH2 1/20 0.33
CES2 O00748 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30872169 0.83 HCRTR2 (0.38) HCRTR2HCRTR1SLC6A7
SCHEMBL31351486 0.82 HCRTR1 (0.56) HCRTR2HCRTR1
SCHEMBL30872179 0.81 PKM (0.38) HCRTR2HCRTR1USP2
SCHEMBL30872180 0.78 HCRTR1 (0.43) HCRTR2HCRTR1EGFR
SCHEMBL30872176 0.76 KDM4E (0.47) HCRTR2HCRTR1ALDH1A1HTTKDM4E
SCHEMBL30872175 0.70 HCRTR1 (0.53) HCRTR2HCRTR1
SCHEMBL30872153 0.68 HCRTR1 (0.56) HCRTR2HCRTR1
SCHEMBL30872161 0.68 HCRTR1 (0.48) HCRTR2HCRTR1
SCHEMBL30872171 0.68 HCRTR1 (0.50) HCRTR2HCRTR1
SCHEMBL30872186 0.67 HCRTR1 (0.45) HCRTR2HCRTR1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024109672-A1 DISUBSTITUTED OCTAHYDROPYRROLO[3,4-C]PYRROLE METHYL KETONE DERIVATIVE AND APPLICATION THEREOF 江苏恩华药业股份有限公司 2024-05-30 WO disclosed