SCHEMBL30877553

SCHEMBL30877553

CCOC(=O)c1nc(C)n2c1CN=C(c1ccccc1F)c1cc(Cl)ccc1-2

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 3/20 0.58
CYP3A4 P08684 2/20 0.58
DRD3 P35462 2/20 0.58
PDE4D Q08499 2/20 0.58
SLC22A1 O15245 1/20 0.58
ABCB11 O95342 1/20 0.58
GABRG2 P18507 3/20 0.55
GABRB3 P28472 3/20 0.55
GABRA3 P34903 2/20 0.55
HTR1A P08908 1/20 0.49
HTR3A P46098 1/20 0.49
KCNH2 Q12809 1/20 0.49
GHSR Q92847 1/20 0.49
TP53 P04637 1/20 0.48
GABRA5 P31644 2/20 0.45
GABRA2 P47869 2/20 0.45
GABRB2 P47870 1/20 0.45
GABRA1 P14867 1/20 0.44
HTR2A P28223 1/20 0.44
ADRA1A P35348 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27185165 1.00 OPRK1 (0.58) OPRK1CYP3A4DRD3PDE4DSLC22A1
SCHEMBL7311633 0.91 GABRG2 (0.54) OPRK1CYP3A4DRD3PDE4DSLC22A1
SCHEMBL7309925 0.91 GABRA3 (0.55) OPRK1CYP3A4DRD3PDE4DSLC22A1
SCHEMBL7313844 0.91 OPRK1 (0.60) OPRK1CYP3A4DRD3PDE4DSLC22A1
SCHEMBL11379951 0.89 OPRK1 (0.57) OPRK1CYP3A4DRD3PDE4DSLC22A1
SCHEMBL5354151 0.88 GABRA2 (0.54) OPRK1GABRG2GABRB3GABRA3KCNH2
SCHEMBL1311112 0.88 OPRK1 (0.63) OPRK1CYP3A4DRD3PDE4DSLC22A1
SCHEMBL7315246 0.88 OPRK1 (0.58) OPRK1CYP3A4DRD3PDE4DSLC22A1
SCHEMBL7317914 0.87 OPRK1 (0.62) OPRK1CYP3A4DRD3PDE4DSLC22A1
SCHEMBL7307575 0.87 GABRG2 (0.62) OPRK1CYP3A4DRD3PDE4DSLC22A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024059669-A2 IMPROVED PROCESS FOR THE PREPARATION OF IMIDAZOBENZODIAZEPINES ODH IP Corp. (US) 2024-03-21 WO disclosed