SCHEMBL30908754

SCHEMBL30908754

CC(C)(C)OC(=O)N[C@@H](CO)C(=O)NCc1ccncc1

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSS P25774 7/20 0.48
CTSK P43235 7/20 0.48
CTSL P07711 1/20 0.48
CTSB P07858 1/20 0.48
BACE1 P56817 8/20 0.47
LMNA P02545 1/20 0.47
MAPT P10636 1/20 0.47
MAPK1 P28482 1/20 0.47
RAB9A P51151 1/20 0.46
CYP17A1 P05093 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29244926 1.00 CTSS (0.48) CTSSCTSKCTSLCTSBBACE1
SCHEMBL30968897 0.87 CTSS (0.62) CTSSCTSKCTSLCTSB
SCHEMBL13583903 0.87 CTSS (0.62) CTSSCTSKCTSLCTSB
SCHEMBL42634 0.87 CTSS (0.62) CTSSCTSKCTSLCTSB
SCHEMBL9582823 0.87 CTSS (0.62) CTSSCTSKCTSLCTSB
SCHEMBL13015865 0.86 PPARG (0.51) CTSSCTSKCTSLCTSB
SCHEMBL993347 0.85 CTSS (0.49) CTSSCTSKCTSLCTSB
SCHEMBL13016479 0.85 CTSS (0.63) CTSSCTSKCTSLCTSBMAPT
SCHEMBL12840932 0.85 CTSS (0.49) CTSSCTSKCTSLCTSB
SCHEMBL7329532 0.82 BACE1 (0.62) CTSSCTSKBACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118055923-A Benzodiazepine derivatives as positive allosteric modulators of the GABAA γ1 receptor 豪夫迈·罗氏有限公司 2024-05-17 CN disclosed