SCHEMBL7329532

SCHEMBL7329532

CC(C)[C@H](NC(=O)OC(C)(C)C)C(=O)NCc1ccncc1

nearest known ligand 0.62

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 17/20 0.62
CTSS P25774 1/20 0.55
CTSK P43235 1/20 0.55
CA2 P00918 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4750042 0.87 CTSS (0.61) BACE1CTSSCTSK
SCHEMBL14102602 0.86 CYP3A4 (0.57) BACE1CTSSCTSKCA2
SCHEMBL8897259 0.86 ALDH1A1 (0.63) BACE1CTSSCTSKCA2
SCHEMBL10276787 0.84 CA2 (0.55) BACE1CTSSCTSKCA2
SCHEMBL10276786 0.84 CA2 (0.55) BACE1CTSSCTSKCA2
SCHEMBL27820614 0.83 CA2 (0.54) BACE1CTSSCTSKCA2
SCHEMBL1752665 0.83 CTSS (0.57) BACE1CTSSCTSKCA2
SCHEMBL30908754 0.82 CTSS (0.48) BACE1CTSSCTSK
SCHEMBL29244926 0.82 CTSS (0.48) BACE1CTSSCTSK
SCHEMBL481947 0.81 RAB9A (0.58)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1990000399-A1 RETROVIRAL PROTEASE BINDING PEPTIDES SMITHKLINE BECKMAN CORPORATION (US) 1990-01-25 WO disclosed
EP-0352000-A2 Retroviral protease binding peptides SMITHKLINE BEECHAM CORPORATION (US) 1990-01-24 EP disclosed