Efloxate

Efloxate

SCHEMBL309159

CCOC(=O)COc1ccc2c(=O)cc(-c3ccccc3)oc2c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 1.00
ALDH1A1 P00352 3/20 0.70
CYP3A4 P08684 2/20 0.70
HPGD P15428 2/20 0.70
CYP1A2 P05177 1/20 0.70
POLB P06746 1/20 0.70
CYP2C9 P11712 1/20 0.70
CYP2C19 P33261 1/20 0.70
MAPT P10636 4/20 0.64
GAA P10253 1/20 0.64
TNKS O95271 2/20 0.60
CYP19A1 P11511 1/20 0.60
SIGMAR1 Q99720 1/20 0.60
NPC1 O15118 1/20 0.60
RAB9A P51151 1/20 0.60
KMT2A Q03164 2/20 0.60
MEN1 O00255 1/20 0.60
LMNA P02545 1/20 0.60
TP53 P04637 1/20 0.60
SMN1; SMN2 Q16637 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11883092 0.86 KDM4E (0.75) KDM4EALDH1A1CYP3A4HPGDCYP1A2
SCHEMBL9141500 0.86 KDM4E (0.74) KDM4EALDH1A1CYP3A4HPGDCYP1A2
SCHEMBL9140701 0.85 KDM4E (0.74) KDM4ECYP3A4CYP1A2MAPTTNKS
SCHEMBL21629622 0.83 ALDH1A1 (0.83) KDM4EALDH1A1HPGDCYP1A2CYP2C19
SCHEMBL8983924 0.82 KDM4E (0.70) KDM4EALDH1A1CYP3A4HPGDCYP1A2
SCHEMBL4053857 0.82 KDM4E (0.80) KDM4EALDH1A1CYP3A4HPGDCYP1A2
SCHEMBL10025659 0.81 SIGMAR1 (0.76) KDM4ECYP3A4MAPTTNKSCYP19A1
SCHEMBL4050048 0.81 KDM4E (0.67) KDM4EALDH1A1CYP3A4HPGDCYP1A2
SCHEMBL10620445 0.80 ALDH1A1 (0.75) KDM4EALDH1A1CYP3A4HPGDCYP1A2
SCHEMBL9139841 0.80 HPGD (0.80) KDM4EALDH1A1CYP3A4HPGDCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1104 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023183932-A2 MONOBODIES BINDING TO INTERCELLULAR ADHESION MOLECULE 2 (ICAM-2) NEW YORK UNIVERSITY (US) 2023-09-28 WO claimed
US-20230093487-A1 VASODILATORS FOR TREATMENT OF HEART FAILURE NORTHEAST OHIO MEDICAL UNIV (US) 2023-03-23 US claimed
EP-4000614-A1 EFLOXATE FOR USE AS ANTIVIRAL AGENT Consejo Superior de Investigaciones Científicas (CSIC) (ES) 2022-05-25 EP claimed
US-11324748-B2 Vasodilators for treatment of heart failure NORTHEAST OHIO MEDICAL UNIVERSITY (US) 2022-05-10 US claimed
EP-3485908-B1 THERAPEUTIC COMBINATION AND USE OF DLL4 ANTAGONIST ANTIBODIES AND ANTI-HYPERTENSIVE AGENTS MEREO BIOPHARMA 5 INC (US) 2021-08-18 EP claimed
US-20200325543-A1 DIAGNOSTIC METHOD TOLREMO THERAPEUTICS AG (CH) 2020-10-15 US claimed
EP-3714069-A1 DIAGNOSTIC METHOD Tolremo Therapeutics AG (CH) 2020-09-30 EP claimed
CN-110128937-A A kind of efficiency light mutagenesis color protective coating 安徽五岳松纳米技术有限公司 2019-08-16 CN claimed
EP-3072526-B1 THERAPEUTIC COMBINATION AND USE OF DLL4 ANTAGONIST ANTIBODIES AND ANTI-HYPERTENSIVE AGENTS ONCOMED PHARM INC (US) 2018-09-26 EP claimed
US-9982042-B2 Therapeutic combination and methods of treatment with a DLL4 antagonist and an anti-hypertensive agent ONCOMED PHARMACEUTICALS, INC. (US) 2018-05-29 US claimed
US-20030162824-A1 Methods of treating or preventing a cardiovascular condition using a cyclooxygenase-1 inhibitor PHARMACIA CORPORATION 2003-08-28 US claimed
WO-2003026705-A1 METHODS FOR STERILIZING BIOLOGICAL MATERIALS USING FLAVONOID/FLAVONOL STABILIZERS CLEARANT, INC. (US) 2003-04-03 WO claimed
US-20030059338-A1 Methods for sterilizing biological materials using flavonoid/flavonol stabilizers CLEARANT, INC. 2003-03-27 US claimed
WO-2002087556-A9 PROBUCOL MONOESTERS AND THEIR USE TO INCREASE PLASMA HDL CHOLESTEROL LEVELS AND IMPROVE HDL FUNCTIONALITY ATHEROGENICS INC (US) 2003-03-20 WO claimed
WO-2002087556-A2 PROBUCOL MONOESTERS AND THEIR USE TO INCREASE PLASMA HDL CHOLESTEROL LEVELS AND IMPROVE HDL FUNCTIONALITY ATHEROGENICS, INC. (US) 2002-11-07 WO claimed
CN-1294519-A Pharmaceutical composition containing a compound having an activity of promoting the absorption of an active ingredient INPHARMA SA (CH) 2001-05-09 CN claimed
EP-1073470-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2001-02-07 EP claimed
WO-2000048636-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2000-08-24 WO claimed
US-5811547-A Method for inducing crystalline state transition in medicinal substance NIPPON SHINYAJU CO., LTD. (JP) 1998-09-22 US claimed
US-5399584-A Preventing gastrointestinal damage caused by nonsteroidal antiinflammatory drugs THE PROCTER & GAMBLE COMPANY (US) 1995-03-21 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230093487-A1 VASODILATORS FOR TREATMENT OF HEART FAILURE VASP, TNNI3, EDNRB KDM4E 4093/4885ALDH1A1 1929/4885CYP3A4 3813/4885
US-20030162824-A1 Methods of treating or preventing a cardiovascular condition using a cyclooxygenase-1 inhibitor PTGS1, PTGIS, TNNT2 KDM4E 4011/4885ALDH1A1 515/4885CYP3A4 867/4885
US-11324748-B2 Vasodilators for treatment of heart failure VASP, TNNI3, EDNRB KDM4E 4093/4885ALDH1A1 1929/4885CYP3A4 3813/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.