SCHEMBL309220

SCHEMBL309220

CCOC(=O)c1cn[nH]c1N

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 1.00
MEN1 O00255 1/20 1.00
KMT2A Q03164 1/20 1.00
TSHR P16473 2/20 0.67
HSD17B10 Q99714 1/20 0.49
NPC1 O15118 5/20 0.48
RAB9A P51151 5/20 0.48
GAA P10253 2/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
HSP90AA1 P07900 1/20 0.47
LMNA P02545 2/20 0.46
KDM4E B2RXH2 2/20 0.46
MAPT P10636 1/20 0.45
HPGD P15428 1/20 0.44
MAPK1 P28482 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28922763 0.85 ALDH1A1 (0.72) ALDH1A1MEN1KMT2ATSHRHSD17B10
SCHEMBL15655280 0.83 ALDH1A1 (0.71) ALDH1A1MEN1KMT2ATSHRHSD17B10
SCHEMBL1420098 0.82 ALDH1A1 (0.70) ALDH1A1MEN1KMT2ATSHRHSD17B10
SCHEMBL20641707 0.81 ALDH1A1 (0.68) ALDH1A1MEN1KMT2ATSHRHSD17B10
SCHEMBL1458672 0.81 ALDH1A1 (0.68) ALDH1A1MEN1KMT2ATSHRHSD17B10
SCHEMBL1009529 0.80 TSHR (1.00) ALDH1A1MEN1KMT2ATSHRHSD17B10
SCHEMBL2324062 0.80 ALDH1A1 (0.67) ALDH1A1MEN1KMT2ATSHRHSD17B10
SCHEMBL25163091 0.79 ALDH1A1 (0.66) ALDH1A1MEN1KMT2ATSHRHSD17B10
SCHEMBL5752771 0.79 ALDH1A1 (0.66) ALDH1A1MEN1KMT2ATSHRHSD17B10
SCHEMBL20303941 0.79 KMT2A (0.66) ALDH1A1MEN1KMT2ATSHRNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 594 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117659025-A TOLL-like receptor 8 (TLR 8) specific antagonists, methods of making and uses thereof 科罗拉多州立大学董事会法人团体 2024-03-08 CN claimed
CN-112110938-A Compound as protein kinase inhibitor and preparation method and application thereof 成都海博为药业有限公司 2020-12-22 CN claimed
CN-111808259-A 3D printing silicone rubber and preparation method and application thereof 四川大学 2020-10-23 CN claimed
CN-110066282-B Pyrazolopyrimidinone compound and preparation method and application thereof 南开大学 2020-07-10 CN claimed
CN-122094678-A AP 2-related kinase 1 inhibitors and uses thereof 2026-05-26 CN disclosed
EP-4724439-A1 HETEROARYL DERIVATIVES AS DDRS INHIBITORS Chiesi Farmaceutici S.p.A. (IT) 2026-04-15 EP disclosed
EP-4725946-A1 IRAK4 DEGRADATION AGENT AND USE THEREOF Guangzhou Unirise Pharmaceutical Co., Ltd. (CN) 2026-04-15 EP disclosed
US-20260070922-A1 PYRAZOLE AND IMIDAZOLE DERIVATIVES AS DUAL OREXIN AND KAPPA-OPIOID RECEPTORS MODULATORS COMPOSITION, METHODS FOR TREATING NEUROLOGICAL AND PSYCHIATRIC DISORDERS HAGER BIOSCIENCES, LLC (US) 2026-03-12 US disclosed
EP-4707276-A2 MALT1 MODULATORS AND USES THEREOF Rarefied Biosciences, Inc. (US) 2026-03-11 EP disclosed
EP-4499611-B1 MALT1 MODULATORS AND USES THEREOF RAREFIED BIOSCIENCES INC (US) 2026-02-18 EP disclosed
EP-4692096-A1 MACROCYCLIC COMPOUND, AND PHARMACEUTICAL COMPOSITION AND USE THEREOF Prime Gene Therapeutics Co., Ltd. (CN) 2026-02-11 EP disclosed
US-20260027217-A1 DEGRADERS THAT TARGET ALK AND THERAPEUTIC USES THEREOF DANA-FARBER CANCER INSTITUTE, INC. (US) 2026-01-29 US disclosed
US-6444696-B1 1-ARYL OR HETEROARYL SUBSTITUTED 5-AMINO-4 CARBONYLPYRAZOLE DERIVATIVES; ANTIINFLAMMATORY AGENTS SYNTEX (U.S.A.) LLC 2002-09-03 US disclosed
US-20020103245-A1 Pyrazole derivatives P38 MAP kinase inhibitors GOLDSTEIN DAVID MICHAEL (US) 2002-08-01 US disclosed
EP-1218346-A1 PYRAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-07-03 EP disclosed
US-6376527-B1 ANTIINFLAMMATORY AGENTS; AUTOIMMUNE DISEASES SYNTEX (U.S.A.) LLC 2002-04-23 US disclosed
US-6316466-B1 Pyrazole derivatives P-38 MAP kinase inhibitors SYNTEX (U.S.A.) LLC 2001-11-13 US disclosed
WO-2001021591-A1 PYRAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2001-03-29 WO disclosed
EP-1075467-A1 PYRAZOLE DERIVATIVES AS P-38 MAP KINASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2001-02-14 EP disclosed
WO-1999057101-A1 PYRAZOLE DERIVATIVES AS P-38 MAP KINASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 1999-11-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260027217-A1 DEGRADERS THAT TARGET ALK AND THERAPEUTIC USES THEREOF ALK, IGF1R, PDGFRB ALDH1A1 855/4885MEN1 2416/4885KMT2A 2199/4885
US-20020103245-A1 Pyrazole derivatives P38 MAP kinase inhibitors MAPK1, MAPK8, MAPKAPK2 ALDH1A1 1667/4885MEN1 4104/4885KMT2A 3772/4885
US-20260070922-A1 PYRAZOLE AND IMIDAZOLE DERIVATIVES AS DUAL OREXIN AND KAPPA-OPIOID RECEPTORS MODULATORS COMPOSITION, METHODS FOR TREATING NEUROLOGICAL AND PSYCHIATRIC DISORDERS OPRK1, OPRD1, HCRTR2 ALDH1A1 1665/4885MEN1 4298/4885KMT2A 1361/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.