SCHEMBL30931995

SCHEMBL30931995

NC(=O)C(=Cc1ccccc1)c1ncccn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C1 Q04828 1/20 0.47
KMT2A Q03164 4/20 0.47
CYP1A2 P05177 2/20 0.47
CYP3A4 P08684 2/20 0.47
CYP2D6 P10635 2/20 0.47
CYP2C9 P11712 2/20 0.47
CYP2C19 P33261 2/20 0.47
MCL1 Q07820 1/20 0.46
MAPT P10636 5/20 0.41
KDM4E B2RXH2 4/20 0.41
ALDH1A1 P00352 4/20 0.41
POLB P06746 3/20 0.41
MAPK1 P28482 2/20 0.41
LMNA P02545 2/20 0.41
MEN1 O00255 2/20 0.41
HPGD P15428 2/20 0.41
HTT P42858 1/20 0.41
NPC1 O15118 6/20 0.40
RAB9A P51151 5/20 0.40
PKM P14618 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21777089 1.00 AKR1C1 (0.47) AKR1C1KMT2ACYP1A2CYP3A4CYP2D6
SCHEMBL23593943 0.77 AKR1C1 (0.70) AKR1C1KMT2ACYP1A2CYP3A4CYP2D6
SCHEMBL2836206 0.77 AKR1C1 (0.70) AKR1C1KMT2ACYP1A2CYP3A4CYP2D6
SCHEMBL6689798 0.77 AKR1C1 (0.70) AKR1C1KMT2ACYP1A2CYP3A4CYP2D6
SCHEMBL16102102 0.77 KMT2A (0.48) AKR1C1KMT2ACYP1A2CYP3A4CYP2D6
SCHEMBL3652897 0.76 NPC1 (0.48) AKR1C1KMT2ACYP1A2CYP3A4CYP2D6
SCHEMBL29979027 0.76 P2RX7 (0.41) KMT2ACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL5014075 0.74 KMT2A (0.38) AKR1C1KMT2ACYP1A2CYP3A4CYP2D6
SCHEMBL16180693 0.73 CYP1A2 (0.55) AKR1C1KMT2ACYP1A2CYP3A4CYP2D6
SCHEMBL20995693 0.71 AKR1C1 (0.43) AKR1C1KMT2ACYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024083111-A1 NOVEL HETEROCYCLIC COMPOUNDS 首药控股(北京)股份有限公司 2024-04-25 WO disclosed