Metamfepramone

Metamfepramone

SCHEMBL309430

CC(C(=O)c1ccccc1)N(C)C

nearest known ligand 0.63

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGR P06401 1/20 0.63
ADRA2A P08913 1/20 0.63
ADRA2B P18089 1/20 0.63
HTR2A P28223 1/20 0.63
HRH1 P35367 1/20 0.63
KCNH2 Q12809 1/20 0.63
RAB9A P51151 3/20 0.50
MAPT P10636 3/20 0.50
NPC1 O15118 2/20 0.50
ATM Q13315 2/20 0.50
HTT P42858 2/20 0.50
MAPK1 P28482 1/20 0.50
NPY5R Q15761 1/20 0.50
LMNA P02545 5/20 0.49
TDP1 Q9NUW8 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
CES2 O00748 1/20 0.47
CES1 P23141 1/20 0.47
ALDH1A1 P00352 4/20 0.44
KDM4E B2RXH2 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Metamfepramone SCHEMBL10505245 1.00 PGR (0.63) PGRADRA2AADRA2BHTR2AHRH1
Metamfepramone SCHEMBL5172661 0.98 PGR (0.61) PGRADRA2AADRA2BHTR2AHRH1
Metamfepramone SCHEMBL22614741 0.98 PGR (0.61) PGRADRA2AADRA2BHTR2AHRH1
SCHEMBL9512907 0.85 HRH1 (0.47) PGRADRA2AADRA2BHTR2AHRH1
SCHEMBL9532923 0.83 PGR (0.59) PGRADRA2AADRA2BHTR2AHRH1
SCHEMBL1223834 0.82 PGR (0.58) PGRADRA2AADRA2BHTR2AHRH1
SCHEMBL15508382 0.81 CA1 (0.47) PGRADRA2AADRA2BHTR2AHRH1
SCHEMBL5954011 0.81 ALDH1A1 (0.48) PGRADRA2AADRA2BHTR2AHRH1
SCHEMBL13813782 0.80 PGR (0.71) PGRADRA2AADRA2BHTR2AHRH1
SCHEMBL29350711 0.80 PGR (0.56) PGRADRA2AADRA2BHTR2AHRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1693 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118184520-A Biphenyl amine compound, preparation method thereof and application thereof in flow battery 中国科学院大连化学物理研究所 2024-06-14 CN claimed
US-20200060997-A1 TARR Receptor Agonists for Sexual Dysfunction JOHN MCCOY 2020-02-27 US claimed
CN-107329368-A A kind of solvable photosensitive composite of alkali and preparation method and application 江苏广信感光新材料股份有限公司 2017-11-07 CN claimed
CN-107203095-A A kind of solvable photosensitive composite of white alkali and preparation method and application 江苏广信感光新材料股份有限公司 2017-09-26 CN claimed
US-20160067271-A1 Methods And Compositions For Preventing Or Treating Obesity NORTHEASTERN UNIVERSITY 2016-03-10 US claimed
US-20150272920-A1 METHOD FOR TREATING OBESITY WITH ANTI-OBESITY FORMULATIONS AND OMEGA 3 FATTY ACIDS FOR THE REDUCTION OF BODY WEIGHT IN CARDIOVASCULAR DISEASE PATIENTS (CVD) AND DIABETICS PIVOTAL THERAPEUTICS INC. (CA) 2015-10-01 US claimed
EP-2814478-A1 A METHOD FOR TREATING OBESITY WITH ANTI-OBESITY FORMULATIONS AND OMEGA 3 FATTY ACIDS FOR THE REDUCTION OF BODY WEIGHT IN CARDIOVASCULAR DISEASE PATIENTS (CVD) AND DIABETICS Pivotal Therapeutics, Inc. (CA) 2014-12-24 EP claimed
US-8715648-B2 Method for treating obesity with anti-obesity formulations and omega 3 fatty acids for the reduction of body weight in cardiovascular disease patients (CVD) and diabetics PIVOTAL THERAPEUTICS INC. (CA) 2014-05-06 US claimed
EP-2675444-A1 A FORMULATIONS COMPRISING OMEGA 3 FATTY ACIDS AND AN ANTI OBESITY AGENT FOR THE REDUCTION OF BODY WEIGHT IN CARDIOVASCULAR DISEASE PATIENTS (CVD) AND DIABETICS Pivotal Therapeutics, Inc. (CA) 2013-12-25 EP claimed
US-20130324461-A1 METHODS AND COMPOSITIONS FOR PREVENTING OR TREATING OBESITY SITKOVSKY MICHAIL V (US) 2013-12-05 US claimed
WO-2003063781-A2 SUBSTITUTED IMIDAZOLES AS CANNABINOID RECEPTOR MODULATORS MERCK & CO., INC. (US) 2003-08-07 WO claimed
US-20030114495-A1 Substituted imidazoles as cannabinoid receptor modulators MERCK SHARP & DOHME CORP. 2003-06-19 US claimed
WO-2003045313-A2 2-AMINOQUINOLINE COMPOUNDS MERCK & CO. INC. (US) 2003-06-05 WO claimed
WO-2003045920-A1 4-AMINOQUINOLINE COMPOUNDS MERCK & CO., INC. (US) 2003-06-05 WO claimed
WO-2003007887-A2 SUBSTITUTED IMIDAZOLES AS CANNABINOID RECEPTOR MODULATORS MERCK & CO., INC. (US) 2003-01-30 WO claimed
JP-2001524960-A 2001-12-04 JP claimed
EP-1073470-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2001-02-07 EP claimed
WO-2000048636-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2000-08-24 WO claimed
EP-0977572-A1 USE OF NK-1 RECEPTOR ANTAGONISTS FOR TREATING EATING DISORDERS MERCK SHARP & DOHME LTD. (GB) 2000-02-09 EP claimed
WO-1998047513-A1 USE OF NK-1 RECEPTOR ANTAGONISTS FOR TREATING EATING DISORDERS MERCK SHARP & DOHME LIMITED (GB) 1998-10-29 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130324461-A1 METHODS AND COMPOSITIONS FOR PREVENTING OR TREATING OBESITY ADORA2A, ADORA3, ADORA1 PGR 2582/4885ADRA2A 16/4885ADRA2B 33/4885
US-20160067271-A1 Methods And Compositions For Preventing Or Treating Obesity ADORA2A, ADORA3, ADORA1 PGR 2582/4885ADRA2A 16/4885ADRA2B 33/4885
US-20030114495-A1 Substituted imidazoles as cannabinoid receptor modulators CNR1, CNR2, GPR119 PGR 2922/4885ADRA2A 426/4885ADRA2B 548/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.