SCHEMBL30944314

SCHEMBL30944314

Cc1cc2nc(NC(=O)C3(C)CCCCC3)sc2c(C)c1Br

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 3/20 0.58
CYP3A4 P08684 2/20 0.45
PI4KB Q9UBF8 1/20 0.45
LCK P06239 1/20 0.41
NPC1 O15118 5/20 0.39
RAB9A P51151 5/20 0.39
KMT2A Q03164 3/20 0.39
MEN1 O00255 2/20 0.39
RXFP1 Q9HBX9 1/20 0.37
HTT P42858 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
CETP P11597 2/20 0.36
ADORA2A P29274 2/20 0.36
P2RX7 Q99572 1/20 0.36
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34
USP21 Q9UK80 1/20 0.34
DYRK1A Q13627 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28523749 0.76 ADORA1 (0.55) ADORA1CYP3A4PI4KBLCKNPC1
SCHEMBL30944326 0.76 ADORA1 (0.55) ADORA1CYP3A4PI4KBLCKNPC1
SCHEMBL30944297 0.76 ADORA1 (0.55) ADORA1CYP3A4PI4KBLCKNPC1
SCHEMBL30944373 0.75 ADORA1 (0.98) ADORA1CYP3A4PI4KBLCKNPC1
SCHEMBL30944341 0.75 ADORA1 (0.80) ADORA1CYP3A4LCKNPC1RAB9A
SCHEMBL30944357 0.75 ADORA1 (0.56) ADORA1CYP3A4PI4KBLCKNPC1
SCHEMBL30944376 0.74 ADORA1 (1.00) ADORA1CYP3A4PI4KBLCKNPC1
SCHEMBL30944352 0.71 DYRK1A (0.63) ADORA1LCKNPC1RAB9AKMT2A
SCHEMBL30944303 0.68 DYRK1A (0.65) ADORA1ADORA2ADYRK1A
SCHEMBL31236382 0.68 DYRK1A (0.65) ADORA1ADORA2ADYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118772080-A Antimycobacterial heterocyclic amides 克莱斯通公司 2024-10-15 CN claimed
CN-118772080-A Antimycobacterial heterocyclic amides 克莱斯通公司 2024-10-15 CN disclosed
CN-112423746-B Novel antimycobacterial heterocyclic amides 克莱斯通公司 2024-06-28 CN disclosed