SCHEMBL30944352

SCHEMBL30944352

CC1(C(=O)Nc2nc3ccc(Cl)cc3s2)CCCCC1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 1/20 0.63
FSCN1 Q16658 1/20 0.63
ADORA1 P30542 1/20 0.63
CASP3 P42574 10/20 0.59
SENP7 Q9BQF6 10/20 0.59
SENP8 Q96LD8 9/20 0.59
SENP6 Q9GZR1 9/20 0.59
CYP2D6 P10635 1/20 0.56
CYP2B6 P20813 1/20 0.56
CYP2C19 P33261 1/20 0.56
LCK P06239 1/20 0.56
NPC1 O15118 5/20 0.55
RAB9A P51151 5/20 0.55
SMN1; SMN2 Q16637 4/20 0.55
KDM4E B2RXH2 3/20 0.55
ALDH1A1 P00352 2/20 0.55
CLK1 P49759 1/20 0.55
PTPN1 P18031 1/20 0.54
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30944341 0.86 ADORA1 (0.80) DYRK1AADORA1CYP2D6CYP2B6CYP2C19
SCHEMBL28518062 0.83 DYRK1A (0.65) DYRK1AADORA1CYP2D6
SCHEMBL30944303 0.83 DYRK1A (0.65) DYRK1AADORA1CYP2D6
SCHEMBL31236382 0.83 DYRK1A (0.65) DYRK1AADORA1CYP2D6
SCHEMBL28527314 0.83 DYRK1A (0.65) DYRK1AADORA1CYP2D6
SCHEMBL30944286 0.82 DYRK1A (0.58) DYRK1AFSCN1CASP3SENP7SENP8
SCHEMBL28512789 0.82 DYRK1A (0.58) DYRK1AFSCN1CASP3SENP7SENP8
SCHEMBL30944362 0.81 DYRK1A (0.67) DYRK1AADORA1CYP2D6
SCHEMBL28519830 0.81 DYRK1A (0.67) DYRK1AADORA1CYP2D6
SCHEMBL30944305 0.81 ADORA1 (0.57) DYRK1AADORA1CYP2C19LCKNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118772080-A Antimycobacterial heterocyclic amides 克莱斯通公司 2024-10-15 CN claimed
CN-118772080-A Antimycobacterial heterocyclic amides 克莱斯通公司 2024-10-15 CN disclosed
CN-112423746-B Novel antimycobacterial heterocyclic amides 克莱斯通公司 2024-06-28 CN disclosed