SCHEMBL30944341

SCHEMBL30944341

CC1(C(=O)Nc2nc3ccc(Br)cc3s2)CCCCC1

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 2/20 0.80
RAB9A P51151 4/20 0.63
NPC1 O15118 3/20 0.63
CYP2C19 P33261 2/20 0.63
DYRK1A Q13627 2/20 0.63
CYP1A2 P05177 1/20 0.63
CYP3A4 P08684 1/20 0.63
CYP2C9 P11712 1/20 0.63
HTT P42858 2/20 0.61
SMN1; SMN2 Q16637 1/20 0.61
CYP2D6 P10635 1/20 0.56
CYP2B6 P20813 1/20 0.56
ALDH1A1 P00352 2/20 0.52
CLK1 P49759 2/20 0.52
TP53 P04637 1/20 0.52
HPGD P15428 1/20 0.52
ADORA2A P29274 1/20 0.51
LCK P06239 1/20 0.51
MAPT P10636 1/20 0.50
LRRK2 Q5S007 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30944373 0.91 ADORA1 (0.98) ADORA1RAB9ANPC1CYP2C19DYRK1A
SCHEMBL30944376 0.89 ADORA1 (1.00) ADORA1RAB9ANPC1CYP2C19DYRK1A
SCHEMBL30944352 0.86 DYRK1A (0.63) ADORA1RAB9ANPC1CYP2C19DYRK1A
SCHEMBL28527314 0.83 DYRK1A (0.65) ADORA1DYRK1ACYP2D6ADORA2ALRRK2
SCHEMBL28518062 0.83 DYRK1A (0.65) ADORA1DYRK1ACYP2D6ADORA2ALRRK2
SCHEMBL30944303 0.83 DYRK1A (0.65) ADORA1DYRK1ACYP2D6ADORA2ALRRK2
SCHEMBL31236382 0.83 DYRK1A (0.65) ADORA1DYRK1ACYP2D6ADORA2ALRRK2
SCHEMBL30944291 0.82 ADORA1 (0.58) ADORA1RAB9ANPC1CYP2C19DYRK1A
SCHEMBL28530522 0.82 ADORA1 (0.58) ADORA1RAB9ANPC1CYP2C19DYRK1A
SCHEMBL30944362 0.81 DYRK1A (0.67) ADORA1DYRK1ACYP2D6ADORA2ALRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118772080-A Antimycobacterial heterocyclic amides 克莱斯通公司 2024-10-15 CN claimed
CN-118772080-A Antimycobacterial heterocyclic amides 克莱斯通公司 2024-10-15 CN disclosed
CN-112423746-B Novel antimycobacterial heterocyclic amides 克莱斯通公司 2024-06-28 CN disclosed