SCHEMBL30965674

SCHEMBL30965674

CC(C)(C)OC(=O)NC1CC2(CCN(CCC3CCN(c4ccc([N+](=O)[O-])cc4F)CC3)CC2)C1

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 9/20 0.55
DRD3 P35462 3/20 0.44
MAPT P10636 5/20 0.41
ALDH1A1 P00352 4/20 0.41
LMNA P02545 3/20 0.41
THRB P10828 1/20 0.40
KMT2A Q03164 2/20 0.39
HTR1A P08908 2/20 0.38
HTR2A P28223 2/20 0.38
MEN1 O00255 1/20 0.38
POLB P06746 1/20 0.38
MAPK1 P28482 1/20 0.38
SLC6A9 P48067 1/20 0.38
SLC6A5 Q9Y345 1/20 0.38
FFAR4 Q5NUL3 1/20 0.38
NAMPT P43490 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30965798 0.89 DRD2 (0.43) DRD2DRD3MAPTALDH1A1LMNA
SCHEMBL29065775 0.89 MAPT (0.47) DRD2MAPTALDH1A1LMNATHRB
SCHEMBL30965765 0.87 MAPT (0.44) DRD2DRD3MAPTALDH1A1LMNA
SCHEMBL30965518 0.87 DRD2 (0.47) DRD2DRD3HTR1AHTR2ANAMPT
SCHEMBL31334849 0.83 DRD2 (0.54) DRD2DRD3MAPTALDH1A1LMNA
SCHEMBL30915181 0.83 DRD2 (0.54) DRD2MAPTALDH1A1LMNATHRB
SCHEMBL13419542 0.83 DRD2 (0.54) DRD2MAPTALDH1A1LMNATHRB
SCHEMBL13419655 0.81 MAPT (0.48) DRD2MAPTALDH1A1LMNATHRB
SCHEMBL30915152 0.81 DRD2 (0.53) DRD2DRD3MAPTALDH1A1LMNA
SCHEMBL31333430 0.81 MAPT (0.51) DRD2MAPTALDH1A1LMNATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4658658-A1 NOVEL PLK1 DEGRADATION INDUCING COMPOUND Uppthera, Inc. (KR) 2025-12-10 EP disclosed
WO-2024162828-A1 NOVEL PLK1 DEGRADATION INDUCING COMPOUND UPPTHERA, INC. (KR) 2024-08-08 WO disclosed