Floredil

Floredil

SCHEMBL309848

CCOc1cc(OCC)cc(OCCN2CCOCC2)c1

nearest known ligand 0.71

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.69
KDM4E B2RXH2 3/20 0.69
HTT P42858 1/20 0.69
MAPK1 P28482 2/20 0.58
CYP1A2 P05177 1/20 0.58
CHRM2 P08172 1/20 0.58
CHRM1 P11229 1/20 0.58
HTR2A P28223 1/20 0.58
SCN1A P35498 1/20 0.58
HTR2B P41595 1/20 0.58
KCNH2 Q12809 1/20 0.58
SCN2A Q99250 1/20 0.58
SIGMAR1 Q99720 1/20 0.58
SCN3A Q9NY46 1/20 0.58
HRH3 Q9Y5N1 1/20 0.58
NPC1 O15118 2/20 0.57
MEN1 O00255 1/20 0.57
KMT2A Q03164 1/20 0.57
USP2 O75604 1/20 0.56
LMNA P02545 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11882168 0.82 KDM4E (0.62) ALDH1A1KDM4EHTTMAPK1CYP1A2
SCHEMBL13107094 0.80 ALDH1A1 (0.73) ALDH1A1KDM4EHTTMAPK1CYP1A2
SCHEMBL15516600 0.80 ALDH1A1 (0.56) ALDH1A1KDM4EHTTMAPK1CYP1A2
SCHEMBL29508217 0.80 ALDH1A1 (0.88) ALDH1A1KDM4EMAPK1CYP1A2CHRM2
SCHEMBL14578276 0.80 ALDH1A1 (0.69) ALDH1A1KDM4EHTTMAPK1NPC1
SCHEMBL7981029 0.80 NPC1 (0.64) ALDH1A1KDM4EMAPK1CYP1A2CHRM2
SCHEMBL13534008 0.79 POLB (0.56) ALDH1A1KDM4EMAPK1CYP1A2CHRM2
SCHEMBL13791665 0.78 MEN1 (0.55) ALDH1A1KDM4EHTTMAPK1CYP1A2
SCHEMBL4306311 0.78 NPC1 (0.49) ALDH1A1KDM4EHTTMAPK1CYP1A2
SCHEMBL4485540 0.78 LTA4H (0.69) ALDH1A1KDM4EMAPK1CYP1A2CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 824 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023183932-A2 MONOBODIES BINDING TO INTERCELLULAR ADHESION MOLECULE 2 (ICAM-2) NEW YORK UNIVERSITY (US) 2023-09-28 WO claimed
US-20230093487-A1 VASODILATORS FOR TREATMENT OF HEART FAILURE NORTHEAST OHIO MEDICAL UNIV (US) 2023-03-23 US claimed
US-11324748-B2 Vasodilators for treatment of heart failure NORTHEAST OHIO MEDICAL UNIVERSITY (US) 2022-05-10 US claimed
EP-3485908-B1 THERAPEUTIC COMBINATION AND USE OF DLL4 ANTAGONIST ANTIBODIES AND ANTI-HYPERTENSIVE AGENTS MEREO BIOPHARMA 5 INC (US) 2021-08-18 EP claimed
EP-3072526-B1 THERAPEUTIC COMBINATION AND USE OF DLL4 ANTAGONIST ANTIBODIES AND ANTI-HYPERTENSIVE AGENTS ONCOMED PHARM INC (US) 2018-09-26 EP claimed
US-9982042-B2 Therapeutic combination and methods of treatment with a DLL4 antagonist and an anti-hypertensive agent ONCOMED PHARMACEUTICALS, INC. (US) 2018-05-29 US claimed
US-20170166632-A1 Therapeutic Combination and Methods of Treatment With A DLL4 Antagonist and an Anti-Hypertensive Agent ONCOMED PHARMACEUTICALS, INC. 2017-06-15 US claimed
US-9511139-B2 Therapeutic combination and methods of treatment with a DLL4 antagonist and an anti-hypertensive agent ONCOMED PHARMACEUTICALS, INC. (US) 2016-12-06 US claimed
EP-3072526-A1 THERAPEUTIC COMBINATION AND USE OF DLL4 ANTAGONIST ANTIBODIES AND ANTI-HYPERTENSIVE AGENTS Oncomed Pharmaceuticals, Inc. (US) 2016-09-28 EP claimed
EP-2488204-B1 THERAPEUTIC COMBINATION AND USE OF DLL4 ANTAGONIST ANTIBODIES AND ANTI-HYPERTENSIVE AGENTS ONCOMED PHARM INC (US) 2016-04-06 EP claimed
WO-2006086544-A2 THERAPEUTIC COMBINATION OF A VEGF ANTAGONIST (VEGF TRAP) AND AN ANTI-HYPERTENSIVE AGENT REGENERON PHARMACEUTICALS, INC. (US) 2006-08-17 WO claimed
EP-1507813-A4 FAT BINDING USING INTER-POLYMER COMPLEX OF GLUCOSAMINE AND POLYACRYLIC ACID RANBAXY LAB LTD (IN) 2005-11-23 EP claimed
EP-1507813-A1 FAT BINDING USING INTER-POLYMER COMPLEX OF GLUCOSAMINE AND POLYACRYLIC ACID Ranbaxy Laboratories Limited (IN) 2005-02-23 EP claimed
EP-1385501-A2 PROBUCOL MONOESTERS AND THEIR USE TO INCREASE PLASMA HDL CHOLESTEROL LEVELS AND IMPROVE HDL FUNCTIONALITY Atherogenics, Inc. (US) 2004-02-04 EP claimed
WO-2003097714-A1 FAT BINDING USING INTER-POLYMER COMPLEX OF GLUCOSAMINE AND POLYACRYLIC ACID RANBAXY LABORATORIES LIMITED (IN) 2003-11-27 WO claimed
US-20030162824-A1 Methods of treating or preventing a cardiovascular condition using a cyclooxygenase-1 inhibitor PHARMACIA CORPORATION 2003-08-28 US claimed
WO-2002087556-A9 PROBUCOL MONOESTERS AND THEIR USE TO INCREASE PLASMA HDL CHOLESTEROL LEVELS AND IMPROVE HDL FUNCTIONALITY ATHEROGENICS INC (US) 2003-03-20 WO claimed
WO-2002087556-A2 PROBUCOL MONOESTERS AND THEIR USE TO INCREASE PLASMA HDL CHOLESTEROL LEVELS AND IMPROVE HDL FUNCTIONALITY ATHEROGENICS, INC. (US) 2002-11-07 WO claimed
EP-1073470-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2001-02-07 EP claimed
WO-2000048636-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2000-08-24 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230093487-A1 VASODILATORS FOR TREATMENT OF HEART FAILURE VASP, TNNI3, EDNRB ALDH1A1 1929/4885KDM4E 4093/4885HTT 2065/4885
US-20030162824-A1 Methods of treating or preventing a cardiovascular condition using a cyclooxygenase-1 inhibitor PTGS1, PTGIS, TNNT2 ALDH1A1 515/4885KDM4E 4011/4885HTT 1804/4885
US-11324748-B2 Vasodilators for treatment of heart failure VASP, TNNI3, EDNRB ALDH1A1 1929/4885KDM4E 4093/4885HTT 2065/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.