SCHEMBL3101

SCHEMBL3101

CCCCS(=O)(=O)N(Cc1ccc(-c2ccccc2C#N)cc1)CC1(C(=O)OCC)CCCCC1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.41
OXTR P30559 2/20 0.38
AVPR1A P37288 2/20 0.38
ITGB1 P05556 1/20 0.36
ITGA4 P13612 1/20 0.36
LTB4R2 Q9NPC1 5/20 0.36
CNR2 P34972 1/20 0.35
FFAR1 O14842 1/20 0.34
AKR1B1 P15121 1/20 0.34
MYC P01106 1/20 0.34
WDR5 P61964 1/20 0.34
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
NR1H4 Q96RI1 1/20 0.33
POLB P06746 1/20 0.33
MME P08473 1/20 0.33
AGTR1 P30556 1/20 0.33
AGTR2 P50052 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2366 0.84 LTB4R2 (0.47) ACHEOXTRAVPR1AITGB1ITGA4
SCHEMBL1911 0.83 LTB4R2 (0.48) ACHEOXTRAVPR1AITGB1ITGA4
SCHEMBL2291 0.82 LTB4R2 (0.35) LTB4R2AGTR1AGTR2
SCHEMBL2563 0.76 ITGB1 (0.42) ACHEOXTRAVPR1AITGB1ITGA4
SCHEMBL8484079 0.75 LTB4R2 (0.40) ACHEOXTRAVPR1AITGB1ITGA4
SCHEMBL2311 0.75 ITGB1 (0.43) ACHEOXTRAVPR1AITGB1ITGA4
SCHEMBL7270209 0.73 LTB4R2 (0.45) ACHEOXTRAVPR1AITGB1ITGA4
SCHEMBL2318 0.72 ACHE (0.44) ACHEOXTRAVPR1AITGB1ITGA4
SCHEMBL2922 0.72 LTB4R2 (0.37) LTB4R2AGTR1AGTR2
SCHEMBL9430039 0.72 LTB4R2 (0.50) ACHEOXTRAVPR1AITGB1ITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0443983-B1 Acyl compounds CIBA GEIGY AG (CH) 1996-02-28 EP disclosed
US-5399578-A Hypotensive; valsartan; high blood pressure and cardiac insufficiency CIBA-GEIGY CORP (US) 1995-03-21 US disclosed
EP-0443983-A1 Acyl compounds CIBA-GEIGY AG (CH) 1991-08-28 EP disclosed