SCHEMBL3105632

SCHEMBL3105632

Fc1ccc(C(Br)c2ccc(Cc3ccc(CBr)cc3)cc2)cc1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 5/20 0.36
TDO2 P48775 2/20 0.36
LOXL2 Q9Y4K0 1/20 0.35
SLC6A2 P23975 2/20 0.35
SLC6A4 P31645 2/20 0.35
SLC6A3 Q01959 2/20 0.35
DAO P14920 1/20 0.35
TAAR1 Q96RJ0 2/20 0.34
TRPA1 O75762 2/20 0.33
ALDH1A1 P00352 1/20 0.33
TSHR P16473 1/20 0.33
HTT P42858 1/20 0.33
AGXT P21549 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3107946 0.82 TRPA1 (0.50) SLC6A2SLC6A4SLC6A3TRPA1ALDH1A1
SCHEMBL3105616 0.82 SLC6A2 (0.37) IDO1SLC6A2SLC6A4SLC6A3TAAR1
SCHEMBL3113885 0.81 KEAP1 (0.38) IDO1DAOTAAR1TRPA1ALDH1A1
SCHEMBL3103451 0.79 IDO1 (0.41) IDO1TDO2LOXL2TAAR1TRPA1
SCHEMBL3111831 0.79 CYP19A1 (0.32) IDO1TDO2SLC6A4SLC6A3DAO
SCHEMBL5110 0.78
SCHEMBL15233233 0.78
SCHEMBL4427290 0.78 IDO1 (0.46) IDO1TDO2SLC6A2SLC6A4SLC6A3
SCHEMBL1835628 0.76 IDO1 (0.50) IDO1LOXL2TAAR1TRPA1ALDH1A1
SCHEMBL22165011 0.76 IDO1 (0.50) IDO1LOXL2TAAR1TRPA1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2163553-B1 ARENE CONNECTED POLYAMINE MACRORING DERIVATIVES, PREPARATION METHODS AND PHARMACEUTICAL USES THEREOF BEIJING MOLECULE SCIENCE AND TECHNOLOGY CO LTD (CN) 2013-12-25 EP disclosed
EP-2163553-A1 ARENE CONNECTED POLYAMINE MACRORING DERIVATIVES, PREPARATION METHODS AND PHARMACEUTICAL USES THEREOF Beijing Molecule Science and Technology Co., Ltd. (CN) 2010-03-17 EP disclosed