SCHEMBL3105616

SCHEMBL3105616

BrCc1ccc(Cc2ccc(C(Br)c3ccc(Br)cc3)cc2)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37
SLC6A3 Q01959 1/20 0.37
TAAR1 Q96RJ0 3/20 0.35
ALDH1A1 P00352 2/20 0.34
TRPA1 O75762 1/20 0.34
TSHR P16473 1/20 0.34
HTR2A P28223 2/20 0.34
HRH3 Q9Y5N1 1/20 0.34
IDO1 P14902 2/20 0.33
HTR1D P28221 1/20 0.33
KDM4E B2RXH2 1/20 0.33
EPHX2 P34913 1/20 0.33
PYCR1 P32322 1/20 0.32
CYP2A6 P11509 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3107946 0.84 TRPA1 (0.50) SLC6A2SLC6A4SLC6A3ALDH1A1TRPA1
SCHEMBL3113885 0.82 KEAP1 (0.38) TAAR1ALDH1A1TRPA1TSHRIDO1
SCHEMBL3105632 0.82 IDO1 (0.36) SLC6A2SLC6A4SLC6A3TAAR1ALDH1A1
SCHEMBL3098973 0.79 ALDH1A1 (0.40) TAAR1ALDH1A1TRPA1TSHRHTR2A
SCHEMBL3103812 0.78 SLC6A2 (0.37) SLC6A2SLC6A4SLC6A3ALDH1A1TRPA1
SCHEMBL7536 0.78
SCHEMBL7187315 0.78 CYP2A6 (0.53) SLC6A2SLC6A4SLC6A3ALDH1A1TSHR
Bromide SCHEMBL29227177 0.75 ALDH1A1 (0.50) TAAR1ALDH1A1TRPA1TSHRHTR2A
SCHEMBL5389732 0.75 ALDH1A1 (0.50) TAAR1ALDH1A1TRPA1TSHRHTR2A
Fluoride SCHEMBL29026731 0.75 ALDH1A1 (0.50) TAAR1ALDH1A1TRPA1TSHRHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2163553-B1 ARENE CONNECTED POLYAMINE MACRORING DERIVATIVES, PREPARATION METHODS AND PHARMACEUTICAL USES THEREOF BEIJING MOLECULE SCIENCE AND TECHNOLOGY CO LTD (CN) 2013-12-25 EP disclosed
EP-2163553-A1 ARENE CONNECTED POLYAMINE MACRORING DERIVATIVES, PREPARATION METHODS AND PHARMACEUTICAL USES THEREOF Beijing Molecule Science and Technology Co., Ltd. (CN) 2010-03-17 EP disclosed